Target Details
| UniProt AC | Q15825 |
|---|---|
| Gene Symbol | CHRNA6 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 92
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (4)
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QWEBUPURHNWVEK
|
7.6 | IC50 | 5 | — | |
ASNYTHIFAFBQFH
|
7.6 | IC50 | 3 | — | |
AQYPBNGIIYVIBQ
|
7.6 | Ki | 5 | — | |
BFESRXFYMDMQQS
|
7.5 | IC50 | 3 | — | |
GPLPNYTYTRIAGH
|
7.5 | IC50 | 3 | — | |
RPQSOKSDYSMFBW
|
7.5 | IC50 | 3 | — | |
JSWKSMHGVJDZBY
|
7.5 | IC50 | 3 | — | |
UPRSNEUCMGKPCF
|
7.4 | IC50 | 3 | — | |
AQYPBNGIIYVIBQ
|
7.4 | Ki | 5 | — | |
QGZBKYBWQCGNTH
|
7.3 | IC50 | 3 | — | |
LVYRPIRSEMMFEE
|
7.3 | IC50 | 3 | — | |
AQYPBNGIIYVIBQ
|
7.3 | Ki | 5 | — | |
AMMQVZPHMBRHME
|
7.2 | IC50 | 3 | — | |
IEYQINPEMQKRDC
|
7.2 | IC50 | 3 | — | |
LKXXWFDWZQRZKV
|
7.2 | IC50 | 3 | — | |
VHTBVZBRBLYBGN
|
7.2 | IC50 | 3 | — | |
XFBDKMSGGGCNAI
|
7.2 | IC50 | 11 | — | |
QAIHOBDHHLOTET
|
7.2 | IC50 | 3 | — | |
VHRLLJQAIUCUDP
|
7.1 | IC50 | 3 | — | |
VXQLPXYMYHKASH
|
7.1 | Ki | 5 | — | |
SNICXCGAKADSCV
|
7.1 | IC50 | 8 | — | |
FAGJOGGAOOMVGD
|
7.1 | IC50 | 3 | — | |
UDMJZFWTHJHTRH
|
7.0 | IC50 | 3 | — | |
INYNWEUTASDACG
|
7.0 | Ki | 5 | — | |
YOWFIQDENDEMRP
|
7.0 | IC50 | 3 | — | |
FANPYQPRSROCKC
|
7.0 | IC50 | 3 | — | |
PRPVVMSCQSOWKN
|
6.9 | IC50 | 3 | — | |
INYNWEUTASDACG
|
6.8 | Ki | 5 | — | |
KMZCUSKKQFNPIY
|
6.7 | Ki | 5 | — | |
VYRZFHOORZTMRI
|
6.7 | IC50 | 3 | — | |
UAFJMITWUKBNEN
|
6.7 | IC50 | 5 | — | |
IBKIPEZDVFQTJT
|
6.6 | Ki | 5 | — | |
LJEPPQATHWQMBV
|
6.6 | Ki | 5 | — | |
IPPNDMWEPHFWFT
|
6.6 | IC50 | 3 | — | |
PWXQAVZNBKKQOF
|
6.5 | Ki | 7 | — | |
INYNWEUTASDACG
|
6.5 | Ki | 5 | — | |
PWXQAVZNBKKQOF
|
6.5 | Ki | 6 | — | |
FIIBHEYGLZGMCK
|
6.5 | Ki | 5 | — | |
AQYPBNGIIYVIBQ
|
6.3 | Ki | 5 | — | |
PKIKIQOOXGRVIT
|
6.2 | Ki | 5 | — | |
NQSGGIDOQYCFCP
|
6.2 | Ki | 5 | — | |
XKGJHXYHHLQEGC
|
6.2 | Ki | 5 | — |