Target Details
| UniProt AC | Q15825 |
|---|---|
| Gene Symbol | CHRNA6 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 92
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (4)
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TUIBLGZTRFZLQY
|
10.2 | Ki | 2 | — | |
RSXPTYRGJDGQJN
|
10.1 | Ki | 2 | — | |
FLAHTCIVXKKZAR
|
9.8 | IC50 | 3 | — | |
GUBZKNSUJVFLNU
|
9.6 | IC50 | 3 | — | |
WHDFCXQEDDAKHI
|
9.6 | IC50 | 3 | — | |
AGSIVKJWYGTAIM
|
9.6 | IC50 | 3 | — | |
QJINNXHOTNMTQO
|
9.4 | Ki | 2 | — | |
QAEMLNYVRDMVAV
|
9.4 | IC50 | 3 | — | |
KGLAXECQSDAPBR
|
9.4 | IC50 | 3 | — | |
FZUKXYWZURLPKR
|
9.3 | Ki | 2 | — | |
YWGWQDYPMLAWGB
|
9.2 | Ki | 2 | — | |
BVYJHUNIDYEALI
|
9.0 | IC50 | 3 | — | |
HOMROBGEZCMEMF
|
9.0 | Ki | 2 | — | |
RCSZDVCUNQPLHO
|
9.0 | Ki | 7 | — | |
BGMUZBOFMKWKCS
|
9.0 | IC50 | 5 | — | |
RCSZDVCUNQPLHO
|
9.0 | Ki | 7 | — | |
PAKVZEJOMQOKAO
|
8.8 | IC50 | 3 | — | |
DUQYFGMBLOPGBY
|
8.8 | IC50 | 3 | — | |
ZUQVZTJFSCBLOT
|
8.8 | IC50 | 3 | — | |
HGIKFFRIFIJEOP
|
8.7 | IC50 | 3 | — | |
SGVSOCSOUHHZAS
|
8.7 | IC50 | 3 | — | |
MXJPOFBPCRQRTD
|
8.7 | IC50 | 3 | — | |
LYGZRGMHPFAAMR
|
8.6 | Ki | 7 | — | |
GLNHQLYIFATJOO
|
8.6 | IC50 | 3 | — | |
HVTMEGQWQQUDIH
|
8.5 | IC50 | 3 | — | |
WYGBFIPJEFIRLV
|
8.5 | IC50 | 3 | — | |
COKJMTQIZQACLZ
|
8.4 | IC50 | 3 | — | |
GTVWKLSULFFQST
|
8.3 | Ki | 7 | — | |
ATDHPNPDBDEQAK
|
8.3 | IC50 | 5 | — | |
WINQUAHGULGZED
|
8.3 | IC50 | 5 | — | |
HQBAWNLKYLZICH
|
8.2 | IC50 | 3 | — | |
VVDRDHLUVVGURR
|
8.2 | IC50 | 5 | — | |
MVQIWKVEEIZQLL
|
8.1 | IC50 | 5 | — | |
YFMOKOLWGKJNCJ
|
8.0 | IC50 | 3 | — | |
AOTZFTGAQIRWOB
|
8.0 | IC50 | 3 | — | |
NMIIKXFGCKOYRV
|
8.0 | IC50 | 5 | — | |
SNXCJPFZRZMRKK
|
8.0 | IC50 | 3 | — | |
DLZUIBOQBIXZPS
|
7.9 | IC50 | 3 | — | |
MFMVYBPYDSNLTE
|
7.9 | IC50 | 3 | — | |
VAPDPQSECMWOFE
|
7.9 | IC50 | 3 | — | |
JTTBYCVBUXQDTE
|
7.9 | IC50 | 3 | — | |
INYNWEUTASDACG
|
7.8 | Ki | 5 | — | |
MLCFZENIQJYRSR
|
7.8 | IC50 | 3 | — | |
DJUPOXJVHQDKPZ
|
7.7 | IC50 | 3 | — | |
QQODMJRPCBCHDU
|
7.7 | IC50 | 3 | — | |
HBRLNTBOOKFZCC
|
7.7 | Ki | 5 | — | |
YJEMXDJGZIOQLT
|
7.7 | IC50 | 3 | — | |
RFCWACSNWRAYNU
|
7.7 | IC50 | 3 | — | |
WXJMNOKWJJRHJY
|
7.7 | IC50 | 3 | — | |
RVUUCOAHJHAFBX
|
7.6 | IC50 | 3 | — |