Target Details
UniProt ACQ15825
Gene SymbolCHRNA6
Protein NameNeuronal acetylcholine receptor subunit alpha-6
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 92
  • Clinical molecules 0
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (92)
InChIKey pChEMBL Type Targets Clinical
TUIBLGZTRFZLQY 10.2 Ki 2
RSXPTYRGJDGQJN 10.1 Ki 2
FLAHTCIVXKKZAR 9.8 IC50 3
GUBZKNSUJVFLNU 9.6 IC50 3
WHDFCXQEDDAKHI 9.6 IC50 3
AGSIVKJWYGTAIM 9.6 IC50 3
QJINNXHOTNMTQO 9.4 Ki 2
QAEMLNYVRDMVAV 9.4 IC50 3
KGLAXECQSDAPBR 9.4 IC50 3
FZUKXYWZURLPKR 9.3 Ki 2
YWGWQDYPMLAWGB 9.2 Ki 2
BVYJHUNIDYEALI 9.0 IC50 3
HOMROBGEZCMEMF 9.0 Ki 2
RCSZDVCUNQPLHO 9.0 Ki 7
BGMUZBOFMKWKCS 9.0 IC50 5
RCSZDVCUNQPLHO 9.0 Ki 7
PAKVZEJOMQOKAO 8.8 IC50 3
DUQYFGMBLOPGBY 8.8 IC50 3
ZUQVZTJFSCBLOT 8.8 IC50 3
HGIKFFRIFIJEOP 8.7 IC50 3
SGVSOCSOUHHZAS 8.7 IC50 3
MXJPOFBPCRQRTD 8.7 IC50 3
LYGZRGMHPFAAMR 8.6 Ki 7
GLNHQLYIFATJOO 8.6 IC50 3
HVTMEGQWQQUDIH 8.5 IC50 3
WYGBFIPJEFIRLV 8.5 IC50 3
COKJMTQIZQACLZ 8.4 IC50 3
GTVWKLSULFFQST 8.3 Ki 7
ATDHPNPDBDEQAK 8.3 IC50 5
WINQUAHGULGZED 8.3 IC50 5
HQBAWNLKYLZICH 8.2 IC50 3
VVDRDHLUVVGURR 8.2 IC50 5
MVQIWKVEEIZQLL 8.1 IC50 5
YFMOKOLWGKJNCJ 8.0 IC50 3
AOTZFTGAQIRWOB 8.0 IC50 3
NMIIKXFGCKOYRV 8.0 IC50 5
SNXCJPFZRZMRKK 8.0 IC50 3
DLZUIBOQBIXZPS 7.9 IC50 3
MFMVYBPYDSNLTE 7.9 IC50 3
VAPDPQSECMWOFE 7.9 IC50 3
JTTBYCVBUXQDTE 7.9 IC50 3
INYNWEUTASDACG 7.8 Ki 5
MLCFZENIQJYRSR 7.8 IC50 3
DJUPOXJVHQDKPZ 7.7 IC50 3
QQODMJRPCBCHDU 7.7 IC50 3
HBRLNTBOOKFZCC 7.7 Ki 5
YJEMXDJGZIOQLT 7.7 IC50 3
RFCWACSNWRAYNU 7.7 IC50 3
WXJMNOKWJJRHJY 7.7 IC50 3
RVUUCOAHJHAFBX 7.6 IC50 3
2D structure