Target Details
| UniProt AC | Q15822 |
|---|---|
| Gene Symbol | CHRNA2 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 24
- Clinical molecules 0
- Avg pChEMBL 8.1
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (24)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QCSHOBIQDLQMMD
|
10.1 | Ki | 3 | — | |
NLPRAJRHRHZCQQ
|
10.0 | Ki | 7 | — | |
JQSHBVHOMNKWFT
|
9.3 | Ki | 6 | — | |
LPYOFVQCAYSFSJ
|
9.1 | IC50 | 6 | — | |
NLPRAJRHRHZCQQ
|
9.0 | Ki | 7 | — | |
UBFPRQOOAXMTBD
|
8.8 | IC50 | 6 | — | |
WONBUILDJNKYCB
|
8.4 | Ki | 5 | — | |
SOEBPVQMXRKIOZ
|
8.3 | Ki | 4 | — | |
SOEBPVQMXRKIOZ
|
8.3 | Ki | 3 | — | |
CCEBJZRLEVFTNS
|
8.1 | Ki | 4 | — | |
CCEBJZRLEVFTNS
|
8.1 | Ki | 3 | — | |
JFPXLNSBLNDHFH
|
8.1 | Ki | 4 | — | |
JFPXLNSBLNDHFH
|
8.1 | Ki | 3 | — | |
MQVPACXYSJDEHQ
|
8.0 | IC50 | 5 | — | |
SNICXCGAKADSCV
|
7.9 | Ki | 5 | — | |
SPTQZFUOJBUHQA
|
7.9 | Ki | 5 | — | |
SPTQZFUOJBUHQA
|
7.9 | Ki | 3 | — | |
TVQVEBXIMQEOQV
|
7.8 | Ki | 4 | — | |
GDXUHGVVRIPSQZ
|
7.5 | Ki | 5 | — | |
SNICXCGAKADSCV
|
7.2 | Ki | 8 | — | |
TVQVEBXIMQEOQV
|
6.9 | Ki | 3 | — | |
CZWUYUYQOZHEAK
|
6.9 | Ki | 3 | — | |
CZWUYUYQOZHEAK
|
6.9 | Ki | 3 | — | |
TVQVEBXIMQEOQV
|
6.0 | Ki | 3 | — |