Target Details
| UniProt AC | Q15750 |
|---|---|
| Gene Symbol | TAB1 |
| Protein Name | TGF-beta-activated kinase 1 and MAP3K7-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00481 (PP2C) |
Summary
- Multi-target molecules 97
- Clinical molecules 1
- Avg pChEMBL 6.87
KEGG Pathways (18)
- Alcoholic liver disease
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Osteoclast differentiation
- Pathogenic Escherichia coli infection
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Yersinia infection
Active Molecules (97)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KJHFJTDIYVBYIY
|
6.5 | IC50 | 2 | — | |
JNOGMCOTCINPDR
|
6.5 | IC50 | 2 | — | |
UEJPPFOPQURDKT
|
6.5 | IC50 | 2 | — | |
WPLBZSRCAZTCEF
|
6.5 | IC50 | 2 | — | |
OQDJNLKOMYTWEB
|
6.5 | IC50 | 2 | — | |
PPDQFCISGDOHIO
|
6.5 | IC50 | 2 | — | |
SUSVWEQZHZXFBT
|
6.5 | IC50 | 2 | — | |
DSQSRIOQMWVLNQ
|
6.5 | IC50 | 2 | — | |
YIGLAOIVUJQLRW
|
6.4 | IC50 | 2 | — | |
NTJCHTSHOGWLTQ
|
6.4 | IC50 | 2 | — | |
OCCSZVQXHVIICH
|
6.4 | IC50 | 2 | — | |
HNRZIHVCJQLPHG
|
6.4 | IC50 | 2 | — | |
NXNILAJGBIVOOD
|
6.4 | IC50 | 2 | — | |
OUAQOOWAHVGVHU
|
6.4 | IC50 | 2 | — | |
UOEIHZWXZHPWMI
|
6.4 | IC50 | 2 | — | |
QNLPTMVMYMACRL
|
6.3 | IC50 | 2 | — | |
NOINHGBAXKOKQW
|
6.3 | IC50 | 2 | — | |
MBDDGSKUZPVINA
|
6.3 | IC50 | 2 | — | |
LDSUSZCVKGCAOW
|
6.3 | IC50 | 2 | — | |
UEJPPFOPQURDKT
|
6.3 | IC50 | 2 | — | |
XESCBULBTJHJDG
|
6.3 | IC50 | 2 | — | |
DNUSNALEWBPUMU
|
6.2 | IC50 | 2 | — | |
RCXJDSKUXDREIO
|
6.2 | IC50 | 2 | — | |
XCKISTZRDFIEIS
|
6.2 | IC50 | 2 | — | |
ZIWQBCKDJZBDIR
|
6.2 | IC50 | 5 | — | |
ZINYHYQBLSXMQW
|
6.2 | IC50 | 2 | — | |
WBVXEKYBEMCCAP
|
6.2 | IC50 | 2 | — | |
JMWLMRFTIKZMEL
|
6.2 | IC50 | 2 | — | |
GMHADLQIMIZPBW
|
6.2 | IC50 | 2 | — | |
KSTJUKWFMNVLEG
|
6.2 | IC50 | 2 | — | |
DFPGPQDBTUYGMY
|
6.1 | IC50 | 2 | — | |
QTEPTJGEVYOFFX
|
6.1 | IC50 | 2 | — | |
LBBOLBNLXHDGBI
|
6.1 | IC50 | 2 | — | |
PNQHSKHLOWEBAN
|
6.1 | IC50 | 2 | — | |
FQVJFULIWJSXIM
|
6.1 | IC50 | 2 | — | |
DBLRPUYTBFIYCV
|
6.1 | IC50 | 2 | — | |
YTNYGYHAAUCRGR
|
6.1 | IC50 | 2 | — | |
CRJDAUAOAIPXJR
|
6.1 | IC50 | 2 | — | |
KKZZPOBLLQUBMJ
|
6.1 | IC50 | 2 | — | |
BKLVJHYYETWJAN
|
6.1 | IC50 | 2 | — | |
KDIQGWYECCPTCS
|
6.1 | IC50 | 2 | — | |
QPZICBYPSUODET
|
6.1 | IC50 | 2 | — | |
LMSVUVDUKNLKGS
|
6.0 | IC50 | 2 | — | |
MVCOAUNKQVWQHZ
|
6.0 | IC50 | 54 | Yes | |
QSGQYRLKAVRIDE
|
6.0 | IC50 | 2 | — | |
CARBIKJGHPINLY
|
6.0 | IC50 | 2 | — | |
PYNBJKLUOZMGRV
|
6.0 | IC50 | 2 | — |