Target Details
| UniProt AC | Q15750 |
|---|---|
| Gene Symbol | TAB1 |
| Protein Name | TGF-beta-activated kinase 1 and MAP3K7-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00481 (PP2C) |
Summary
- Multi-target molecules 97
- Clinical molecules 1
- Avg pChEMBL 6.87
KEGG Pathways (18)
- Alcoholic liver disease
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Osteoclast differentiation
- Pathogenic Escherichia coli infection
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Yersinia infection
Active Molecules (97)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QEAYKBGEHPZBIL
|
8.7 | IC50 | 2 | — | |
RNDSPZADISTGBT
|
8.5 | IC50 | 2 | — | |
XDCWLOMVUOZXFY
|
8.4 | IC50 | 2 | — | |
JURMELNKITYBRM
|
8.4 | IC50 | 2 | — | |
YQZZHUQLRWPXNZ
|
8.4 | IC50 | 2 | — | |
JTCXCSWNNQIPRO
|
8.3 | IC50 | 2 | — | |
FVFLNMVKWNRXOS
|
8.3 | IC50 | 2 | — | |
ZQACLJMUNJMDKP
|
8.2 | IC50 | 2 | — | |
VZWXALUQDOYOJQ
|
8.1 | IC50 | 2 | — | |
NEQZWEXWOFPKOT
|
8.1 | IC50 | 9 | — | |
WFHQLAWBICSWPO
|
8.1 | IC50 | 4 | — | |
OIZYRHLPFJOIQM
|
7.9 | IC50 | 2 | — | |
UNYPOOKIBOGJII
|
7.9 | IC50 | 2 | — | |
CQMWAJCVQYHQCJ
|
7.8 | IC50 | 2 | — | |
IIBQLYSZHMEQIH
|
7.8 | IC50 | 2 | — | |
IXXBWYJJOYSCNJ
|
7.8 | IC50 | 2 | — | |
VLSKNLVBBCEHSR
|
7.8 | IC50 | 2 | — | |
VGAICDJDNKCITB
|
7.8 | IC50 | 2 | — | |
PZPZZBSXXDLNMN
|
7.7 | IC50 | 2 | — | |
HREDYOVSBYDONU
|
7.6 | IC50 | 2 | — | |
MJJJFOLDERHCND
|
7.5 | IC50 | 2 | — | |
SSNQAUBBJYCSMY
|
7.5 | IC50 | 5 | — | |
ZWXIOQDBSVHEGC
|
7.5 | IC50 | 2 | — | |
QWDMOLLUOYFWOV
|
7.5 | IC50 | 3 | — | |
BKXGJUGZEFIAJO
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 408 | — | |
LEVZCGPPIDIGHW
|
7.4 | IC50 | 2 | — | |
HUFPFCSZVXOFRZ
|
7.4 | IC50 | 2 | — | |
RQFOIAOPEILIMX
|
7.4 | IC50 | 2 | — | |
KFTLSWHJVMUFGV
|
7.3 | IC50 | 2 | — | |
YYTVWIMHEXZBKS
|
7.2 | IC50 | 2 | — | |
LSSSBVSRWFCJKB
|
7.1 | IC50 | 2 | — | |
IHXGKMUEVBBWBZ
|
7.0 | IC50 | 2 | — | |
OMSUAZHPXSYOQO
|
7.0 | IC50 | 2 | — | |
XGQCOOMJAUFAOT
|
7.0 | IC50 | 2 | — | |
LTQRMOSYFBRQRH
|
7.0 | IC50 | 2 | — | |
JXNXZCJQWOEXJV
|
6.9 | IC50 | 2 | — | |
UPJJRELFFCGJGA
|
6.8 | IC50 | 2 | — | |
RUNVBUSNWGRNAS
|
6.8 | IC50 | 2 | — | |
PCGJEVAVUOYIQB
|
6.8 | IC50 | 2 | — | |
SPEMUMBPRQTTAA
|
6.8 | IC50 | 2 | — | |
FFTUIKFDUYMWTI
|
6.8 | IC50 | 5 | — | |
NTUWMPKGQOZJLQ
|
6.8 | IC50 | 2 | — | |
FCYFQTBWJKSDFR
|
6.7 | IC50 | 2 | — | |
YSMQCLKSRAHMMV
|
6.7 | IC50 | 2 | — | |
SPEMUMBPRQTTAA
|
6.7 | IC50 | 2 | — | |
FJPOGNAHCZFDQR
|
6.6 | IC50 | 2 | — | |
PXVURKNFXLGXEF
|
6.6 | IC50 | 2 | — | |
QMKZTPJYKZRXJU
|
6.6 | IC50 | 2 | — | |
QZUXSJFGHNXNFE
|
6.6 | IC50 | 2 | — |