Target Details
| UniProt AC | Q15746 |
|---|---|
| Gene Symbol | MYLK |
| Protein Name | Myosin light chain kinase, smooth muscle |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16620 (23ISL) PF00041 (fn3) PF07679 (I-set) PF00069 (Pkinase) |
Summary
- Multi-target molecules 42
- Clinical molecules 13
- Avg pChEMBL 6.84
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
9.5 | Kd | 1075 | — | |
FYSRKRZDBHOFAY
|
8.5 | Kd | 8 | — | |
HZTYDQRUAWIZRE
|
8.0 | Kd | 40 | Yes | |
UIARLYUEJFELEN
|
7.9 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
GDVRVPIXWXOKQO
|
7.8 | IC50 | 10 | — | |
KOZFSFOOLUUIGY
|
7.8 | Ki | 26 | — | |
KOZFSFOOLUUIGY
|
7.7 | IC50 | 88 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | IC50 | 408 | — | |
KOZFSFOOLUUIGY
|
7.6 | IC50 | 15 | Yes | |
ZBNZXTGUTAYRHI
|
7.1 | Kd | 102 | Yes | |
LNMRSSIMGCDUTP
|
7.1 | Kd | 13 | — | |
XQVVPGYIWAGRNI
|
7.0 | Kd | 34 | — | |
PHXJVRSECIGDHY
|
7.0 | Kd | 59 | — | |
AXWDQRXGOKDXJT
|
6.8 | Kd | 6 | — | |
QDLHCMPXEPAAMD
|
6.8 | IC50 | 13 | Yes | |
ZCCPLJOKGAACRT
|
6.7 | Kd | 599 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
DORZPJWJOBMQKC
|
6.6 | IC50 | 9 | — | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
CZWJLLBPWLUINU
|
6.5 | IC50 | 10 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
HFNKQEVNSGCOJV
|
6.4 | Kd | 65 | — | |
NXSJMRCTGYTSTK
|
6.4 | Kd | 200 | — | |
CVWXJKQAOSCOAB
|
6.4 | Kd | 35 | — | |
UBPYILGKFZZVDX
|
6.3 | Kd | 130 | Yes | |
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
WULUGQONDYDNKY
|
6.3 | IC50 | 5 | — | |
GUBJNPWVIUFSTR
|
6.2 | Kd | 103 | — | |
JMWUINDPNXOLQK
|
6.2 | Ki | 2 | — | |
NJRSAZRJYRWJJH
|
6.2 | Ki | 2 | — | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
BPNUQXPIQBZCMR
|
6.1 | Kd | 83 | Yes | |
GMZCYCKIXQZORP
|
6.0 | IC50 | 6 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |