Target Details
UniProt ACQ15661
Gene SymbolTPSAB1
Protein NameTryptase alpha/beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 342
  • Clinical molecules 0
  • Avg pChEMBL 7.63
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (342)
InChIKey pChEMBL Type Targets Clinical
DUGSEPGMXTZBQB 6.8 IC50 4
DUQNWFHMCCTXDR 6.8 Ki 2
QZKOOEFIMWKZPK 6.8 Ki 9
XQGVJTLGUGOPAJ 6.8 Ki 5
LLHQEYJISFCOIX 6.8 IC50 4
ICJRTFAHVMZUFX 6.8 Ki 2
NLDZDRVLDYNPMO 6.8 Ki 4
SLMWQRNSGOARMV 6.8 Ki 2
MMYBWDFBCFGBTQ 6.8 IC50 3
JFOWLBVJJJQNFR 6.8 Ki 2
RFJQDANCBUZHLP 6.8 IC50 3
YKBINVNRXCQAQH 6.8 IC50 4
FOGVEVTZPZCRAO 6.8 Ki 3
GWDQDTYXFJAZKY 6.8 Ki 4
UUIRCTHWPGTOIL 6.8 Ki 2
ZAICATAUIFLGRH 6.8 Ki 3
DQCDHYDRHXLVIM 6.7 Ki 2
AMLUFTPKUZYFEG 6.7 IC50 4
AXAWARWVQYJXEC 6.7 IC50 2
OSPQCZJJZMQHLM 6.7 IC50 4
GDGRKBROPOHQAC 6.7 Ki 2
FVIQCYPEJUJZQG 6.7 IC50 2
XLHDYTQMNPVLMS 6.7 IC50 4
GJNNFTSDQAHBMY 6.7 IC50 2
OGNWJRBFZUEUEW 6.7 Ki 4
SDQBWRWAMSSQIA 6.7 Ki 3
YWBAIBRDVBWQDN 6.7 IC50 4
JMUOMUDAWFHUPQ 6.7 Ki 5
POKLRFBZRALDRW 6.6 IC50 4
VYBUDYVARMKISV 6.6 Ki 5
DCRMWXPALBAKDE 6.6 Ki 3
XNZOSJOWGGIDEH 6.6 Ki 2
ZSAGRGVSQBYUNU 6.6 Ki 2
NUHSLCPNNDENLB 6.6 Ki 4
SQJJYHFSTOCHPK 6.6 IC50 4
WOCBHXLMEDMERT 6.6 IC50 3
QCOWDIVJHRGAHU 6.6 IC50 2
BIESPJYZQAPZAA 6.5 IC50 4
MQGBZTPKIUNIBN 6.5 Ki 2
UPTLBLRIQLXTMC 6.5 Ki 2
KBGIRKZCBHNGJB 6.5 Ki 2
KDLUBAQRBALVKK 6.5 Ki 4
ZXBRUEFMBNYVGU 6.5 Ki 3
LINNHGYRJMKPGT 6.5 Ki 2
SKYWIMYOGAWOMB 6.5 Ki 2
DFFMTKSEWMVESR 6.5 Ki 2
COXCETVPGDANPN 6.5 Ki 2
HEZYHVJSUKHORA 6.5 IC50 3
IBXHKTQHOKLBOK 6.5 IC50 3
PCLFVAAOFXTGFD 6.5 IC50 3
2D structure