Target Details
UniProt ACQ15661
Gene SymbolTPSAB1
Protein NameTryptase alpha/beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 342
  • Clinical molecules 0
  • Avg pChEMBL 7.63
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (342)
InChIKey pChEMBL Type Targets Clinical
USPWLAOSWVJNQB 8.2 IC50 3
WYGJQXPPZGICFJ 8.2 IC50 4
ZPTYDNODWOJNDO 8.2 IC50 4
ZWNQLNNVHMLKBK 8.2 IC50 4
HGTDLVZISKJFRC 8.2 Ki 2
DDPNTOHALTYXKV 8.2 Ki 5
QRBIRSCLEVEODD 8.2 Ki 4
LIEHLGBNHWHLEQ 8.2 Ki 2
OXLOPODZLRDMRO 8.2 Ki 5
VUINSGHDSKJJIY 8.2 Ki 4
ASVJMKPNFKPPKC 8.2 IC50 3
AUYOZPJOPWTGLF 8.2 IC50 4
HFMJHADXPOTJRL 8.2 IC50 4
QHEOSDZWICETJC 8.1 Ki 3
ZFODODBXWGBNAV 8.1 Ki 5
FACNOXIVXQYGTJ 8.1 Ki 4
BGGZHUZBDMWKHC 8.1 IC50 3
MAEITLFHBBOJEY 8.1 Ki 4
MIGYGQICECQJBG 8.1 Ki 2
MRKOFZIYRYJJKV 8.1 IC50 3
PZPGGBJAZPANHC 8.1 IC50 4
XCWCBDGDVLDSNP 8.1 IC50 3
FHXAHHBOZHKKNJ 8.0 Ki 2
WISAGRHYXNSVKU 8.0 Ki 5
DOSXWQFAKWWFPY 8.0 Ki 5
ANCMGNKVWBLMLM 8.0 Ki 3
CUNHNEOCSUHSFO 8.0 Ki 4
FHSYWSNXYHJDBM 8.0 IC50 4
MWWOPUUDOBRJOT 8.0 Ki 2
UUELGVPSDQEDNK 8.0 Ki 5
IPPCSGWUBIZOOZ 8.0 Ki 5
LCFBXXJFKDZQHQ 8.0 IC50 3
MWDTYWNRQRBAGQ 8.0 Ki 5
PHDVQHYFNDKHCG 8.0 Ki 2
UHKBIDYPVMVONS 8.0 Ki 4
MBUXHFXIOHKMBL 7.9 IC50 3
VYXQZBSQSKQRJB 7.9 Ki 5
WCCFVFLUYLVNMZ 7.9 IC50 4
KLDNWEHWZPDGQL 7.9 Ki 4
OSOVTHSUTDEIKI 7.9 IC50 4
VOHBOBKPRLGZFP 7.9 Ki 5
ZCBOGFQZYMUMCO 7.9 IC50 3
MUMKNKHFNSSKED 7.8 Ki 4
TUUQUGIFKQSJSD 7.8 IC50 4
VXDAVYUFYPFGDX 7.8 Ki 5
ITSMYKQDPHZPSC 7.8 IC50 4
BCYMMXPTRFITIK 7.8 Ki 4
IJSFLTKQJAUFSB 7.8 Ki 4
JFGPIRSKQQLIBV 7.8 Ki 4
MBBNKWIBPSNEBE 7.8 Ki 5
2D structure