Target Details
UniProt ACQ15661
Gene SymbolTPSAB1
Protein NameTryptase alpha/beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 342
  • Clinical molecules 0
  • Avg pChEMBL 7.63
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (342)
InChIKey pChEMBL Type Targets Clinical
ZEDMSBVBKUUZHF 8.7 IC50 4
IPZMZRVZLGSWFC 8.7 Ki 5
GJGQMDQFASCGME 8.6 Ki 5
WMMQSAVOXZFUEI 8.6 Ki 5
PWHBUXLKTXHYAP 8.6 Ki 5
HRGUCUMYYOYQMA 8.5 Ki 5
MLWLRPHVDMLHHG 8.5 Ki 5
CYOAJSVBGQTLDM 8.5 Ki 4
FIYVZQGLSZYNFI 8.5 IC50 3
PJXUQCYMECYEFS 8.5 Ki 3
PKWZPPLXHJULQB 8.5 Ki 2
PTNWHYHSUZCKAD 8.5 Ki 5
ACIRAJIHJQLJDI 8.5 Ki 2
ZAXACLDYKLBPPT 8.5 Ki 5
ZRTJJNYEQYCQHW 8.5 Ki 5
FYOXGAYJIRAPBZ 8.4 Ki 5
CTQGEVXMPHYTEG 8.4 Ki 5
QXNONEMELKQESX 8.4 Ki 5
WLLZIGJHUQLYKB 8.4 Ki 5
GVMXAPWPASJXDG 8.4 Ki 3
HJGSVTBWNGCVCA 8.4 IC50 3
MBMPSQUPSWCBFW 8.4 Ki 3
MFTQITSPGQORDA 8.4 IC50 9
PUWISFZBZKJLMA 8.4 Ki 3
RFLIXMUMFBXMBJ 8.4 IC50 4
TZJAJXIWPGHOCJ 8.4 IC50 3
YFBRXKLPGVWRRC 8.4 Ki 4
NQUQNMFOLYWMAE 8.3 IC50 3
ZYDNPDIXLNZESB 8.3 Ki 2
JFCVNWMMGCAHDT 8.3 Ki 5
ABNTXKAUVWBRSK 8.3 IC50 3
ACULTQKPVQHRLM 8.3 Ki 2
FQRONIICHHLFKW 8.3 IC50 4
ILGKFMNQEJFIGC 8.3 Ki 4
JLFJBLLDESQVDQ 8.3 Ki 2
MFKKOBLWAUMGNF 8.3 IC50 2
PHUOJJOCYCBHRI 8.3 IC50 3
QVNABSFZNDQTGX 8.3 IC50 4
RTVGVVNPBUBPDD 8.3 IC50 4
SVZDUPPWBBYATM 8.3 Ki 5
VUCRJVPKFXYFDP 8.3 IC50 4
WURLDWQYIPYVLC 8.3 IC50 4
XBZOJHFKWCFSLM 8.3 Ki 5
WKMOUBHSDIPQLZ 8.3 IC50 3
PQVCEZVKPWHTFF 8.3 Ki 6
DUHWZEZYOPJXCS 8.2 Ki 2
NGEVXLYYUCTKSC 8.2 Ki 5
RFFVSYIMXSVIFA 8.2 Ki 5
SEFDHSMOCPXWGA 8.2 Ki 4
LYDBHSDWPNKPJD 8.2 IC50 4
2D structure