Target Details
UniProt ACQ15661
Gene SymbolTPSAB1
Protein NameTryptase alpha/beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00089 (Trypsin)
Summary
  • Multi-target molecules 342
  • Clinical molecules 0
  • Avg pChEMBL 7.63
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (342)
InChIKey pChEMBL Type Targets Clinical
YQZZYTVUJVKJSN 10.7 Ki 4
ALVVXKNOSDJRDJ 10.6 Ki 4
RRBKNHHBEVRVIE 10.5 Ki 4
PODYAQNNRUPOOJ 10.3 Ki 4
XBLJTWKIPZEWCV 10.2 Ki 4
BYQFZIDMWZQLEL 10.2 Ki 4
MYOWXFMSAIUPOT 10.0 Ki 4
NLJGWVWBVAVMER 10.0 Ki 3
VYZARPYDAFKXDL 9.9 Ki 4
MGVGXPSFFJZQMX 9.7 Ki 4
CBGNIBUPSHCBIU 9.4 IC50 3
SZSTYZLOARLHRK 9.4 Ki 4
WCTYMQLNWCHQSB 9.4 Ki 3
WKPLTJYUKCBVTC 9.4 Ki 5
XLCNADMNCIGXSS 9.4 Ki 3
BJUPAZWABXENNS 9.3 Ki 4
SCBIPCJXEMVPQX 9.3 Ki 3
UKPPUXUTDBVVBU 9.3 Ki 3
IEDBGWNXIHURPN 9.2 Ki 4
HXHUFCTVAIQYDR 9.2 IC50 3
IXQBHQLSEXDXIE 9.2 IC50 3
OSOWUTPJQXFFRX 9.2 Ki 3
QGIQDOYBACRUDW 9.1 Ki 4
HMISKNUPRCAHAW 9.0 Ki 4
BOPGBYFJKNADGK 9.0 IC50 6
CQOOFDORTITLOU 9.0 IC50 3
DBMMRUFZHANFAD 9.0 IC50 3
FXPVOGVCAKWEON 9.0 IC50 4
FYVVIEIXYWNGDL 9.0 IC50 5
LSNAYDZARICVGA 9.0 IC50 4
OAIOSQMKFBSMMD 9.0 Ki 4
OSMZQODSQZAXHL 9.0 IC50 3
VRWYRMFZKQAXPQ 9.0 IC50 4
AZEBDSIKGXLILJ 9.0 Ki 4
UGTQPXSJRSGZSL 8.9 Ki 4
FSYLSIDSZSXSDO 8.9 Ki 2
LPBADDHUZIZZHC 8.8 Ki 2
QIHKHBGQSKPTOB 8.8 Ki 5
FHCQLMSOTXBNCN 8.8 IC50 4
RFHHWPRQNRHMMZ 8.8 Ki 5
ZTETUVWDHVYMFI 8.8 Ki 5
CSXORICIIMOCOR 8.7 Ki 5
KFSSZEQPFJUGTN 8.7 Ki 5
XVYFBYVSZOCXRJ 8.7 IC50 4
FAPNFKWYERZNCS 8.7 Ki 5
OUFUAGQUIQUBPV 8.7 IC50 3
PGTIPBIHTMRPEQ 8.7 Ki 5
BYOZXEFJRSCZIK 8.7 Ki 4
VMPGWEWOIGDNDK 8.7 Ki 5
XLQCDKFBSFWDOO 8.7 Ki 4
2D structure