Target Details
| UniProt AC | Q15569 |
|---|---|
| Gene Symbol | TESK1 |
| Protein Name | Dual specificity testis-specific protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 14
- Clinical molecules 4
- Avg pChEMBL 6.83
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
10.1 | Kd | 599 | — | |
ZBNZXTGUTAYRHI
|
7.5 | Kd | 102 | Yes | |
VAARYSWULJUGST
|
7.1 | Kd | 119 | Yes | |
SEJGTFPOEJWEGG
|
6.6 | Kd | 149 | — | |
CXQHYVUVSFXTMY
|
6.6 | Kd | 154 | — | |
HKSZLNNOFSGOKW
|
6.6 | IC50 | 408 | — | |
UIARLYUEJFELEN
|
6.5 | Kd | 289 | Yes | |
UQRCJCNVNUFYDX
|
6.5 | Kd | 27 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
HKSZLNNOFSGOKW
|
6.5 | Kd | 213 | — | |
NHHQJBCNYHBUSI
|
6.4 | Kd | 220 | — | |
KTEIFNKAUNYNJU
|
6.4 | Kd | 114 | — | |
WUCYRTXFXRZKSV
|
6.3 | IC50 | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |