Target Details
| UniProt AC | Q15562 |
|---|---|
| Gene Symbol | TEAD2 |
| Protein Name | Transcriptional enhancer factor TEF-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01285 (TEA) PF17725 (YBD) |
Summary
- Multi-target molecules 180
- Clinical molecules 0
- Avg pChEMBL 7.1
KEGG Pathways (3)
Active Molecules (180)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTCVDVMTUCELSN
|
8.7 | IC50 | 4 | — | |
OVIHDIFRRBKOFL
|
8.5 | IC50 | 4 | — | |
CEAPHBAEPGSQPT
|
8.5 | IC50 | 4 | — | |
DOJLPEPHMDZDEC
|
8.5 | IC50 | 4 | — | |
OLEOCPIYXWADHD
|
8.5 | IC50 | 4 | — | |
GKNRLFKBMBYKNY
|
8.5 | IC50 | 4 | — | |
HJZNAABVSQNGNB
|
8.5 | IC50 | 4 | — | |
PRTRRNCTFDDRTL
|
8.4 | IC50 | 4 | — | |
FATYKAPPXHGOKR
|
8.4 | IC50 | 4 | — | |
MAALNNWDTHSDCS
|
8.4 | IC50 | 4 | — | |
QTORWETWLFGNQW
|
8.4 | IC50 | 4 | — | |
LZVAGKBBWFBYJU
|
8.3 | IC50 | 4 | — | |
XXBTVYDNQBOFDF
|
8.3 | IC50 | 4 | — | |
WDCQVSJMVAYRHG
|
8.2 | IC50 | 4 | — | |
XRRQRUDVKCNHSM
|
8.2 | IC50 | 4 | — | |
AFCYMBUDPUSDIK
|
8.2 | IC50 | 4 | — | |
JRNWBFIHIFCYKC
|
8.2 | IC50 | 4 | — | |
LZVAGKBBWFBYJU
|
8.2 | IC50 | 4 | — | |
NCICSHLFRCFOTN
|
8.1 | IC50 | 4 | — | |
XRRQRUDVKCNHSM
|
8.1 | IC50 | 4 | — | |
LZINKSRQWFTLRX
|
8.1 | IC50 | 4 | — | |
JVDHMGGKKVAVRQ
|
8.1 | IC50 | 4 | — | |
LZINKSRQWFTLRX
|
8.1 | IC50 | 4 | — | |
KQRNWDALNMUUOG
|
8.1 | IC50 | 4 | — | |
HFIXCQZNBIBHKU
|
8.1 | IC50 | 4 | — | |
GKNRLFKBMBYKNY
|
8.0 | IC50 | 4 | — | |
GXCQIZYKYRQWBI
|
8.0 | IC50 | 4 | — | |
MRLLZKOSLONRSI
|
8.0 | IC50 | 5 | — | |
KNYXOZFGQRNBDN
|
7.9 | IC50 | 4 | — | |
MAFUTVMOVXZBEL
|
7.8 | IC50 | 4 | — | |
OWLSOTDTUQFGNX
|
7.8 | IC50 | 4 | — | |
WDCQVSJMVAYRHG
|
7.8 | IC50 | 3 | — | |
OTGMINCKHGEJQA
|
7.8 | IC50 | 4 | — | |
IAVQMKDYNYOXGY
|
7.7 | IC50 | 3 | — | |
UVLIYPUDQMULNH
|
7.7 | IC50 | 4 | — | |
XXBTVYDNQBOFDF
|
7.7 | IC50 | 4 | — | |
PWQJFURIOYPGCQ
|
7.6 | IC50 | 4 | — | |
FLMGNCNJKWNPAH
|
7.6 | IC50 | 4 | — | |
UKVLFZYWLKTJHR
|
7.6 | IC50 | 4 | — | |
KXCKTSLTRHZBEF
|
7.6 | IC50 | 4 | — | |
MEGPPIOBIKDGEA
|
7.6 | IC50 | 4 | — | |
SRCSMFOAKKIMCL
|
7.6 | IC50 | 4 | — | |
MAFUTVMOVXZBEL
|
7.5 | IC50 | 4 | — | |
JXOOXNVSLKJZEL
|
7.5 | IC50 | 4 | — | |
DJGXOJSWOLDZPW
|
7.5 | IC50 | 4 | — | |
NEZOBPSNSLEAJQ
|
7.5 | IC50 | 4 | — | |
NCICSHLFRCFOTN
|
7.5 | IC50 | 4 | — | |
JVDHMGGKKVAVRQ
|
7.5 | IC50 | 4 | — | |
AAYVOUUBHRKCMZ
|
7.5 | IC50 | 4 | — | |
WLQCJPPBRDDTTG
|
7.4 | IC50 | 3 | — |