Target Details
| UniProt AC | Q15418 |
|---|---|
| Gene Symbol | RPS6KA1 |
| Protein Name | Ribosomal protein S6 kinase alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 144
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (10)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJIAQDJKSXQLIT
|
6.7 | Kd | 38 | — | |
AOKADEMCVOQECP
|
6.6 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
6.6 | Kd | 112 | — | |
UBGKZPSSXPFLIM
|
6.6 | IC50 | 2 | — | |
WABHLXQVOYVYTI
|
6.6 | IC50 | 3 | — | |
GPXKVULNYYNGDP
|
6.5 | IC50 | 4 | — | |
UEJXELMBDCXXAQ
|
6.5 | IC50 | 9 | — | |
CDMGBJANTYXAIV
|
6.5 | Kd | 34 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
AXTAPYRUEKNRBA
|
6.5 | IC50 | 24 | — | |
YBYYWUUUGCNAHQ
|
6.4 | IC50 | 8 | — | |
KZYAHEIPPAPADQ
|
6.4 | IC50 | 3 | — | |
UHTHHESEBZOYNR
|
6.4 | Kd | 66 | Yes | |
ZCBUQCWBWNUWSU
|
6.4 | Kd | 59 | — | |
HZTYDQRUAWIZRE
|
6.4 | Kd | 40 | Yes | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
LOLPPWBBNUVNQZ
|
6.3 | Kd | 97 | Yes | |
QDULKFTXPAMMHU
|
6.3 | IC50 | 2 | — | |
QQJKCGXOHWHBQV
|
6.3 | IC50 | 4 | — | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
XMRDIROQMJMYRD
|
6.3 | IC50 | 4 | — | |
YHFGSBURESFKPZ
|
6.3 | IC50 | 4 | — | |
GEWPHZNCWUIEEN
|
6.3 | IC50 | 3 | — | |
JZRNXAPRPJTGOG
|
6.3 | Kd | 3 | — | |
QRULDXBXPXGMQS
|
6.2 | IC50 | 3 | — | |
YHVHYWYQEFELOW
|
6.2 | IC50 | 44 | — | |
QMGUOJYZJKLOLH
|
6.2 | IC50 | 21 | Yes | |
RHTXWIKPNGROHZ
|
6.2 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
UFJUPXKMZSBZPZ
|
6.2 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.1 | Kd | 82 | Yes | |
PDSGDBHQLRAVID
|
6.1 | IC50 | 2 | — | |
PALTUSLCLFDFQQ
|
6.1 | IC50 | 9 | — | |
OLIIUAHHAZEXEX
|
6.1 | IC50 | 3 | — | |
SOUYYRXENUITFU
|
6.1 | IC50 | 2 | — | |
FLBNLJLONKAPLR
|
6.1 | Kd | 31 | — | |
KWQTWTSUJDYVIO
|
6.1 | IC50 | 5 | — | |
MCBPNFWHHNJTGN
|
6.1 | IC50 | 5 | — | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
HWTKDUIKACSTLX
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |