Target Details
| UniProt AC | Q15418 |
|---|---|
| Gene Symbol | RPS6KA1 |
| Protein Name | Ribosomal protein S6 kinase alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 144
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (10)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDDDPIGPOLUCED
|
7.8 | IC50 | 2 | — | |
KMVDGCBYEJXIME
|
7.8 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
SDLDUDKFDXGWAV
|
7.8 | IC50 | 4 | — | |
LKHWQSZVOZRQIZ
|
7.8 | IC50 | 4 | — | |
JAUXVEYDNKFQJQ
|
7.7 | IC50 | 2 | — | |
XIYKGCYSJCRNDN
|
7.7 | IC50 | 4 | — | |
DWRUMXZDNGCUDK
|
7.6 | IC50 | 3 | — | |
XYMNFMNOEWBPNB
|
7.6 | IC50 | 4 | — | |
UGHABJRZQKZAHP
|
7.6 | IC50 | 6 | — | |
LHNSCZROXVKHFK
|
7.6 | IC50 | 3 | — | |
RSFBRAHCHZGZPB
|
7.5 | IC50 | 8 | — | |
AILRADAXUVEEIR
|
7.5 | IC50 | 75 | — | |
ZIJDDQGSYWWTTP
|
7.5 | IC50 | 2 | — | |
DTEKTGDVSARYDS
|
7.5 | IC50 | 11 | — | |
CXSQMXRQOZZFLD
|
7.5 | IC50 | 18 | — | |
IIRWNGPLJQXWFJ
|
7.5 | IC50 | 21 | — | |
PHWHNHYZZNJPLB
|
7.5 | IC50 | 6 | Yes | |
KYVBBJIEKCCZTM
|
7.4 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
WRSGIHWQWREBIP
|
7.4 | IC50 | 2 | — | |
OAYXVYXQZWJEBE
|
7.4 | IC50 | 4 | — | |
YDELNSXADYPQGS
|
7.3 | IC50 | 15 | Yes | |
CZIVUSJISIAXJB
|
7.3 | IC50 | 18 | — | |
AYCPARAPKDAOEN
|
7.3 | IC50 | 73 | — | |
LAJAFFLJAJMYLK
|
7.2 | IC50 | 17 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
FBECJFYYKBIJPC
|
7.2 | IC50 | 2 | — | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
SXRCGQAHDJRHJC
|
7.2 | IC50 | 4 | — | |
YVQOYBIBWBAHKH
|
7.1 | IC50 | 12 | — | |
OYNBTBJATZVIGH
|
7.0 | IC50 | 3 | — | |
SXOZSDJHGMAEGZ
|
7.0 | IC50 | 2 | — | |
QDIMOURDMVMOHZ
|
7.0 | IC50 | 3 | — | |
HBDSHCUSXQATPO
|
7.0 | IC50 | 14 | Yes | |
HIUHVDROHDSKTC
|
7.0 | Ki | 20 | — | |
IBRKIEOOAVIRDE
|
7.0 | IC50 | 2 | — | |
JCSGFHVFHSKIJH
|
7.0 | IC50 | 10 | Yes | |
HFNKQEVNSGCOJV
|
6.9 | Kd | 65 | — | |
SXDPQGRNHSLZPC
|
6.9 | IC50 | 18 | — | |
YOVNFNXUCOWYSG
|
6.9 | IC50 | 33 | Yes | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
WVXNSAVVKYZVOE
|
6.8 | IC50 | 92 | — | |
MBCJUIJWPYUEBX
|
6.8 | IC50 | 7 | — | |
QHKYPYXTTXKZST
|
6.8 | Kd | 28 | — | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
DSXXEELGXBCYNQ
|
6.7 | IC50 | 28 | Yes | |
XHBVYDAKJHETMP
|
6.7 | IC50 | 24 | Yes | |
JRKYKAKARRYSSS
|
6.7 | IC50 | 14 | Yes |