Target Details
| UniProt AC | Q15418 |
|---|---|
| Gene Symbol | RPS6KA1 |
| Protein Name | Ribosomal protein S6 kinase alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 144
- Clinical molecules 20
- Avg pChEMBL 7.41
KEGG Pathways (10)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YISMQBFJYDFMAL
|
9.7 | IC50 | 46 | — | |
HKSZLNNOFSGOKW
|
9.7 | IC50 | 408 | — | |
ZIIWGJMMDJWIKB
|
9.7 | IC50 | 7 | — | |
HVOCYKRGXDBAPR
|
9.4 | IC50 | 3 | — | |
JOMGWMSWUXJNHR
|
9.3 | IC50 | 3 | — | |
PAOJZRPLNNXONF
|
9.3 | IC50 | 3 | — | |
MTAFDCDGNPHAKS
|
9.2 | IC50 | 3 | — | |
ZASQNOFKMXADOA
|
9.2 | IC50 | 3 | — | |
SENHYTFMMJPFHA
|
9.2 | IC50 | 3 | — | |
LWLOLQIXHMFYND
|
9.0 | IC50 | 3 | — | |
MXSRCGHETGMNGI
|
9.0 | IC50 | 3 | — | |
XJSPSRRPVKOQCW
|
9.0 | IC50 | 3 | — | |
FNPBMTZGHSTSCD
|
8.8 | IC50 | 3 | — | |
JXSXWPCGHMFVGR
|
8.8 | IC50 | 3 | — | |
PCZMIWZARLASMT
|
8.8 | IC50 | 2 | — | |
NNEGEHDJOHHIGP
|
8.7 | IC50 | 3 | — | |
VANVVQOKOBHKMX
|
8.7 | IC50 | 2 | — | |
AIZHXUUSVDWSRD
|
8.7 | IC50 | 3 | — | |
XMJMYXPPWSLYBN
|
8.6 | IC50 | 3 | — | |
AXONTVKFBHBALT
|
8.6 | IC50 | 3 | — | |
HWENSJQGPPXSPG
|
8.5 | IC50 | 3 | — | |
RJHWXUSDSADOOD
|
8.5 | IC50 | 3 | — | |
LKHWQSZVOZRQIZ
|
8.4 | IC50 | 6 | — | |
QWHJEDGXVYDZGR
|
8.4 | IC50 | 3 | — | |
BWNZRZRECKJDGL
|
8.4 | IC50 | 3 | — | |
LVLFSSZNAIKYCD
|
8.4 | IC50 | 19 | — | |
XGVWHMVZYCTASP
|
8.4 | IC50 | 3 | — | |
BWGRHTJKFKCSGW
|
8.3 | IC50 | 3 | — | |
ZCITXZXBLWIHHP
|
8.3 | IC50 | 6 | — | |
XEZNMDMVOXPEQL
|
8.3 | IC50 | 3 | — | |
CGECJCJUHCZZGO
|
8.3 | IC50 | 9 | — | |
UXYSSMZFOQFSRB
|
8.3 | IC50 | 2 | — | |
YUYJEQHNWKQNBT
|
8.3 | IC50 | 3 | — | |
MACWQTHSUCWPOE
|
8.2 | IC50 | 3 | — | |
BNYVNKCEEQZWJL
|
8.2 | IC50 | 3 | — | |
IKUFKDGKRLMXEX
|
8.2 | IC50 | 3 | — | |
JNQOAFHFWORJSO
|
8.2 | IC50 | 2 | — | |
RJCVQFMGMSMVAX
|
8.2 | IC50 | 3 | — | |
FYXRSVDHGLUMHB
|
8.2 | IC50 | 8 | — | |
ZMXMTLXHUISIRF
|
8.1 | IC50 | 3 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
NBCDCMYRULBOTN
|
8.1 | IC50 | 3 | — | |
LKHWQSZVOZRQIZ
|
8.1 | IC50 | 4 | — | |
PQBOEVFVXNDSJY
|
8.1 | IC50 | 2 | — | |
OZFFKOSQNBBYCA
|
8.0 | IC50 | 12 | — | |
VKEHHFHLZFTOGI
|
8.0 | IC50 | 2 | — | |
RYTILZIKFSZLNP
|
8.0 | IC50 | 2 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
NXXSVEQIIURRGX
|
7.9 | IC50 | 3 | — | |
CJROUFPGIGKBGZ
|
7.8 | IC50 | 3 | — |