Target Details
| UniProt AC | Q15375 |
|---|---|
| Gene Symbol | EPHA7 |
| Protein Name | Ephrin type-A receptor 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 41
- Clinical molecules 14
- Avg pChEMBL 6.79
KEGG Pathways (1)
Active Molecules (41)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YOBIWCLAYQWPPW
|
8.8 | IC50 | 23 | — | |
CXQHYVUVSFXTMY
|
8.4 | Kd | 154 | — | |
SUXYGJZMCWKJJI
|
8.4 | IC50 | 26 | Yes | |
LOLPPWBBNUVNQZ
|
8.1 | Kd | 97 | Yes | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — | |
ALKJNCZNEOTEMP
|
7.8 | Kd | 55 | — | |
HVXKQKFEHMGHSL
|
7.7 | Kd | 21 | — | |
XKFTZKGMDDZMJI
|
7.4 | Kd | 64 | Yes | |
UHTHHESEBZOYNR
|
7.3 | Kd | 66 | Yes | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
UQRCJCNVNUFYDX
|
7.1 | Kd | 27 | — | |
WVXNSAVVKYZVOE
|
7.1 | IC50 | 92 | — | |
MPVGZUGXCQEXTM
|
7.0 | Kd | 61 | Yes | |
YHVHYWYQEFELOW
|
6.8 | IC50 | 44 | — | |
BGQOUQWQPRPBKN
|
6.8 | IC50 | 7 | — | |
APPXQUDJLJXULP
|
6.7 | IC50 | 47 | — | |
IUGBGEUCXVKGQK
|
6.7 | Kd | 13 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
WPXVVAWAHQHJPF
|
6.7 | IC50 | 41 | — | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
OMZCMEYTWSXEPZ
|
6.6 | Kd | 43 | Yes | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
HKSZLNNOFSGOKW
|
6.4 | Kd | 213 | — | |
AAKJLRGGTJKAMG
|
6.4 | Kd | 50 | Yes | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
RAHBGWKEPAQNFF
|
6.3 | Kd | 26 | — | |
XGALLCVXEZPNRQ
|
6.2 | Kd | 39 | Yes | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
XXJWYDDUDKYVKI
|
6.2 | Kd | 52 | — | |
IRPVABHDSJVBNZ
|
6.2 | IC50 | 6 | — | |
MLDQJTXFUGDVEO
|
6.2 | Kd | 85 | Yes | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
NXSJMRCTGYTSTK
|
6.1 | Kd | 200 | — | |
MVCOAUNKQVWQHZ
|
6.1 | Kd | 54 | Yes | |
OSVUGUHRKMMBSE
|
6.0 | Kd | 170 | — | |
HHFBDROWDBDFBR
|
6.0 | Kd | 40 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |