Target Details
| UniProt AC | Q15349 |
|---|---|
| Gene Symbol | RPS6KA2 |
| Protein Name | Ribosomal protein S6 kinase alpha-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 109
- Clinical molecules 10
- Avg pChEMBL 7.28
KEGG Pathways (10)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FMGZGKDQXIZQLF
|
6.1 | IC50 | 2 | — | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
ZVYLAQPDMUKXOT
|
6.1 | IC50 | 5 | — | |
HIUHVDROHDSKTC
|
6.0 | Ki | 20 | — | |
KCVOKHWVSRPHJC
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
XDOILUADECHLAS
|
6.0 | IC50 | 2 | — |