Target Details
| UniProt AC | Q15349 |
|---|---|
| Gene Symbol | RPS6KA2 |
| Protein Name | Ribosomal protein S6 kinase alpha-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 109
- Clinical molecules 10
- Avg pChEMBL 7.28
KEGG Pathways (10)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWXDZAYQHRBBQT
|
7.4 | IC50 | 2 | — | |
PIPGGBLVUJYMED
|
7.4 | IC50 | 3 | — | |
ZQMGSEHFOOINGT
|
7.4 | IC50 | 2 | — | |
WXEZWMNXEPCNCY
|
7.4 | IC50 | 2 | — | |
ULNZFQKAFXCYBO
|
7.4 | IC50 | 2 | — | |
FOLSZCLZVLICGG
|
7.3 | IC50 | 2 | — | |
HFTWWDARPWZARK
|
7.3 | IC50 | 3 | — | |
LCVZRKFDNWPBET
|
7.3 | IC50 | 2 | — | |
CHFKZEPYDHGBQK
|
7.3 | IC50 | 2 | — | |
LZAHKCVOJMJNFW
|
7.3 | IC50 | 2 | — | |
WDXXELAFEZBSNE
|
7.3 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
YARFNYLGLQVPEB
|
7.2 | IC50 | 2 | — | |
YVQOYBIBWBAHKH
|
7.2 | IC50 | 12 | — | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
JSFCBYKENXVGRL
|
7.2 | IC50 | 2 | — | |
WBSLEWFFUMKPFM
|
7.2 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
UERCXNOQFSTSOY
|
7.1 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
CPDJVFPDCVMFHF
|
7.0 | IC50 | 2 | — | |
XYMNFMNOEWBPNB
|
7.0 | IC50 | 4 | — | |
HFNKQEVNSGCOJV
|
6.8 | Kd | 65 | — | |
GMVUXANRAYNFHC
|
6.7 | IC50 | 2 | — | |
WGAAHZPAINDSDB
|
6.7 | IC50 | 2 | — | |
AATRJMCVLUZFSH
|
6.7 | IC50 | 2 | — | |
AXRCEOKUDYDWLF
|
6.7 | Kd | 31 | — | |
FLSKMXCIDGMHDI
|
6.7 | IC50 | 2 | — | |
LHRDCIRKYUFYOY
|
6.7 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
BTCGJYJHCYOBJS
|
6.6 | IC50 | 2 | — | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
NMSKCMQPIFOSHU
|
6.5 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.5 | Kd | 137 | Yes | |
OTMPGQSHVZZPJK
|
6.5 | IC50 | 2 | — | |
XEMRFXZAJHTFCF
|
6.4 | IC50 | 2 | — | |
JRNJNYBQQYBCLE
|
6.4 | Kd | 40 | Yes | |
LUYLGHWQUPWABZ
|
6.4 | IC50 | 2 | — | |
KDKUVYLMPJIGKA
|
6.4 | Kd | 91 | Yes | |
ZNPMPVBLJKHNSN
|
6.4 | IC50 | 2 | — | |
FCTSFXREUIQMDP
|
6.4 | IC50 | 2 | — | |
BFIIPSNMXRZJOY
|
6.3 | IC50 | 2 | — | |
BGACUNRYWOIUJH
|
6.3 | IC50 | 2 | — | |
VVEBCQLECIQGHE
|
6.2 | IC50 | 2 | — | |
UJLAWZDWDVHWOW
|
6.2 | Kd | 16 | — | |
LRHLPBFCDHGQOT
|
6.2 | IC50 | 2 | — | |
YMKXWFUPUHDFKL
|
6.2 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
XQVVPGYIWAGRNI
|
6.2 | Kd | 34 | — | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes |