Target Details
| UniProt AC | Q15349 |
|---|---|
| Gene Symbol | RPS6KA2 |
| Protein Name | Ribosomal protein S6 kinase alpha-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 109
- Clinical molecules 10
- Avg pChEMBL 7.28
KEGG Pathways (10)
Active Molecules (109)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LOLPPWBBNUVNQZ
|
9.0 | IC50 | 97 | Yes | |
NRGYMIVHSWOTKI
|
9.0 | IC50 | 2 | — | |
ZHMXXVNQAFCXKK
|
9.0 | IC50 | 15 | — | |
WKUUMSASAHOWGZ
|
8.7 | IC50 | 2 | — | |
BRBMDFAROPPCNO
|
8.5 | IC50 | 2 | — | |
IKUFKDGKRLMXEX
|
8.4 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
8.4 | Kd | 170 | — | |
ZWUCWBYYVLQXEP
|
8.4 | IC50 | 4 | — | |
TWQIEMARYWIEFU
|
8.4 | IC50 | 2 | — | |
WMGGYIKBPUVPFM
|
8.4 | IC50 | 2 | — | |
XVKPIWUWUZOHIR
|
8.2 | IC50 | 3 | — | |
QQXZJQAEELFYDV
|
8.2 | IC50 | 2 | — | |
FYXRSVDHGLUMHB
|
8.2 | IC50 | 8 | — | |
LAJAFFLJAJMYLK
|
8.2 | IC50 | 17 | — | |
YUYJEQHNWKQNBT
|
8.1 | IC50 | 3 | — | |
YVUHNKZPGGBYDH
|
8.1 | IC50 | 2 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
NXSJMRCTGYTSTK
|
8.1 | Kd | 200 | — | |
HKSZLNNOFSGOKW
|
8.1 | Kd | 408 | — | |
WIICYVHPNFINMO
|
8.1 | IC50 | 2 | — | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
QHBRARNRIAKCGO
|
8.0 | IC50 | 2 | — | |
XECUHDNZTMADFD
|
8.0 | IC50 | 2 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
AYCPARAPKDAOEN
|
8.0 | Ki | 73 | — | |
PXRIUZVVLPVSSH
|
8.0 | IC50 | 2 | — | |
IIRWNGPLJQXWFJ
|
7.9 | IC50 | 21 | — | |
QYLAYPRSSJNQDC
|
7.9 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
7.9 | IC50 | 75 | — | |
ZHMXXVNQAFCXKK
|
7.8 | IC50 | 2 | — | |
YEOMJKKERMIQSA
|
7.8 | IC50 | 2 | — | |
DTEKTGDVSARYDS
|
7.8 | IC50 | 11 | — | |
UJAUSTYSRUCHNY
|
7.7 | IC50 | 2 | — | |
SPOWSXDVDODVEW
|
7.7 | IC50 | 2 | — | |
HZZNLCVNOOMGDD
|
7.7 | IC50 | 2 | — | |
VCZQSUBZCZZLAX
|
7.7 | IC50 | 2 | — | |
XRTXYXCNVWUOKB
|
7.7 | IC50 | 2 | — | |
ZDYXRELDNKSUBF
|
7.7 | IC50 | 2 | — | |
KAKNBLVUBRXYQD
|
7.7 | IC50 | 2 | — | |
UTARVXNWFXWXPH
|
7.7 | IC50 | 2 | — | |
BRBMDFAROPPCNO
|
7.7 | IC50 | 2 | — | |
OZFFKOSQNBBYCA
|
7.6 | IC50 | 12 | — | |
LQERXZYSNKIMFN
|
7.6 | IC50 | 2 | — | |
VSYFECVWSJTEIL
|
7.6 | IC50 | 2 | — | |
JBOKTWNEIMBJNQ
|
7.6 | IC50 | 2 | — | |
LQZKYXLZCLMOGP
|
7.6 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
RSFBRAHCHZGZPB
|
7.5 | IC50 | 8 | — | |
MVRDTJDXYOJXNF
|
7.5 | IC50 | 2 | — | |
FTOWCRNOCYACIS
|
7.4 | IC50 | 2 | — |