Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNTCGRJDUJEUDG
|
6.2 | Ki | 37 | — | |
CXDUFDRGOOEEHL
|
6.2 | IC50 | 3 | — | |
IZAVTOABECKIDH
|
6.2 | Ki | 20 | — | |
JCUNURGXJBYRFK
|
6.2 | IC50 | 3 | Yes | |
NRZYTPAJGVTKIM
|
6.2 | Ki | 38 | — | |
RTDSHUGNRVXRHN
|
6.2 | Ki | 51 | — | |
UMGYMAXDIGYRMA
|
6.2 | IC50 | 3 | — | |
XBYVOPRDASFDMY
|
6.2 | Ki | 42 | — | |
MCIZZPUSTVXXPG
|
6.2 | IC50 | 3 | Yes | |
OKYKKFLCZPGQHI
|
6.2 | IC50 | 5 | — | |
DLCOHYNRTMTHQE
|
6.2 | IC50 | 2 | — | |
QLFTUFXDFRRBKL
|
6.2 | IC50 | 2 | — | |
CJAOTOWETHYRND
|
6.1 | IC50 | 5 | — | |
GJDYHVMPMKOHGG
|
6.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 213 | — | |
CFIBXVQLBVNOHW
|
6.1 | Ki | 64 | — | |
MSSFKFFUKSRZMQ
|
6.1 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
6.1 | Kd | 170 | — | |
PQNWNVWJXPSZFR
|
6.1 | Ki | 21 | — | |
SKBWQUPLWQUWPH
|
6.1 | IC50 | 6 | Yes | |
SGQJPPQXKVUHGS
|
6.1 | IC50 | 6 | Yes | |
HGYLDYXQKAISMX
|
6.0 | Kd | 4 | — | |
KPZGJWPPVXZLDN
|
6.0 | IC50 | 10 | — | |
FEPYBAFFXFFSLC
|
6.0 | IC50 | 3 | — | |
VAARYSWULJUGST
|
6.0 | Kd | 119 | Yes | |
CTJAMSGCMYAVCZ
|
6.0 | Ki | 14 | — | |
GXJSLIOOPZRPEV
|
6.0 | Ki | 34 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KOHNRDPXFDZZJF
|
6.0 | Ki | 31 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OSAWFUCUZJNEID
|
6.0 | IC50 | 20 | — | |
OWFXKTOLFUQPDJ
|
6.0 | Ki | 36 | — | |
SEJLPXCPMNSRAM
|
6.0 | IC50 | 7 | — | |
VOXXNSOMSGHJJR
|
6.0 | Ki | 3 | — | |
ZCCJKVBTHCOISJ
|
6.0 | Ki | 46 | — |