Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MDTJFOFYNXHTKV
|
6.6 | IC50 | 5 | — | |
AQAMLFJHLGJOCZ
|
6.6 | IC50 | 5 | — | |
QGZVSVHWQCGWDX
|
6.6 | IC50 | 3 | — | |
ZYQXEVJIFYIBHZ
|
6.6 | IC50 | 5 | — | |
JCKPXXCMARLTQI
|
6.6 | IC50 | 6 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
NKUFCHJXONJOLU
|
6.5 | IC50 | 4 | — | |
VIVGTLWPQZQFPV
|
6.5 | IC50 | 2 | — | |
IYCITBYBDPSBBJ
|
6.5 | IC50 | 6 | — | |
QSGIGRAFESHIBA
|
6.5 | IC50 | 3 | — | |
FQGVUAQWOXXERW
|
6.5 | IC50 | 3 | Yes | |
PAFOOYBINUNMGT
|
6.5 | IC50 | 6 | Yes | |
MNXBPMHJGAAMCB
|
6.5 | IC50 | 2 | — | |
XZAATUBTUPPERZ
|
6.5 | IC50 | 6 | — | |
VEUPQFZZGZKGQD
|
6.5 | IC50 | 3 | — | |
DYWKHZDUSFUFCP
|
6.4 | IC50 | 3 | — | |
LWXXXBLCUHRMAR
|
6.4 | IC50 | 3 | — | |
LXURGGKEOPHREO
|
6.4 | IC50 | 13 | — | |
VXJXHNMYRAHBBO
|
6.4 | IC50 | 5 | — | |
DLQXAWIVHRHOQT
|
6.4 | IC50 | 6 | Yes | |
CQXFMKMVOOUGSS
|
6.4 | Ki | 6 | — | |
GCBJDOWIQHMCMR
|
6.4 | Ki | 84 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
XSGCQHSBQMZVQA
|
6.4 | IC50 | 2 | — | |
CMFVTAHMZDUCJB
|
6.4 | IC50 | 10 | — | |
DWJSVGCODPLRLP
|
6.4 | IC50 | 3 | — | |
XGALLCVXEZPNRQ
|
6.4 | IC50 | 39 | Yes | |
XILHUDGNEDEXFJ
|
6.4 | IC50 | 3 | — | |
XPUIECRALWERTL
|
6.4 | IC50 | 4 | — | |
YUEWCBSNZWDONI
|
6.3 | IC50 | 3 | — | |
QYZOGCMHVIGURT
|
6.3 | Kd | 26 | Yes | |
UHTHHESEBZOYNR
|
6.3 | Kd | 66 | Yes | |
DIYFLUKUTVHJCO
|
6.3 | IC50 | 3 | — | |
BIKYDWLMTPRSQL
|
6.3 | Ki | 50 | — | |
NXSJMRCTGYTSTK
|
6.3 | Kd | 200 | — | |
PKCDDUHJAFVJJB
|
6.3 | Ki | 13 | — | |
RQVKVJIRFKVPBF
|
6.3 | Ki | 13 | — | |
XHORJSJFHVABEA
|
6.3 | Ki | 49 | — | |
YEHCNYAQEBQCCS
|
6.3 | Ki | 74 | — | |
YMIJUBCSOKSFRU
|
6.3 | Ki | 87 | — | |
DJCDHWXQLRMRTB
|
6.3 | IC50 | 5 | — | |
WDTHDWKPTWWHLS
|
6.3 | IC50 | 13 | — | |
FYSLYZBOZFMTDD
|
6.3 | IC50 | 6 | Yes | |
AYNLVZLZOVZSHL
|
6.3 | IC50 | 3 | — | |
QAWQPXUVEVTPDR
|
6.3 | IC50 | 3 | — | |
IZUCNCXKMINXNV
|
6.2 | IC50 | 4 | — | |
ZCNCSRRXBRIFQF
|
6.2 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
CXQHYVUVSFXTMY
|
6.2 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.2 | Kd | 149 | — |