Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXFGHUNNGNQSMQ
|
7.0 | Ki | 19 | — | |
LDLBFITVAGVRNV
|
7.0 | IC50 | 6 | Yes | |
SBRIQINKAOKMMM
|
7.0 | IC50 | 6 | — | |
ZKHDDJKHTPLPOQ
|
7.0 | Ki | 62 | — | |
AHONPWLSTJWLMC
|
7.0 | IC50 | 3 | — | |
SGQJPPQXKVUHGS
|
7.0 | IC50 | 6 | Yes | |
ALLOGFWHFYNGAI
|
7.0 | IC50 | 4 | — | |
ZXNLHZGFHDHRCO
|
7.0 | IC50 | 4 | — | |
YSROCLXNQLJIKL
|
7.0 | IC50 | 5 | — | |
AHBFBRPGNOVEBK
|
6.9 | IC50 | 11 | — | |
YHVHYWYQEFELOW
|
6.9 | IC50 | 44 | — | |
MVJMMLFMPWITEJ
|
6.9 | Ki | 110 | — | |
ZVWRFVCNQOECJS
|
6.9 | Ki | 71 | — | |
RGZXAQQHXALOBL
|
6.9 | Kd | 10 | — | |
WVUNYSQLFKLYNI
|
6.9 | IC50 | 46 | Yes | |
ALZWUAVTIXIKIX
|
6.9 | IC50 | 3 | — | |
SKFDSQFYKXYVPS
|
6.8 | IC50 | 9 | Yes | |
YMQSEEOAYCTNQU
|
6.8 | IC50 | 3 | — | |
JEQABWAFHZXXLZ
|
6.8 | IC50 | 4 | — | |
LJQVSABKPVFCTG
|
6.8 | IC50 | 4 | — | |
LVNYQEFSHJDOCT
|
6.8 | IC50 | 4 | — | |
QCJFYACTZIVZBB
|
6.8 | IC50 | 8 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
HYCYVMNKZFALHN
|
6.8 | IC50 | 5 | — | |
ICDUDMAKDBBZOT
|
6.8 | IC50 | 3 | — | |
YRMOQCDUODUCRH
|
6.8 | IC50 | 3 | — | |
OMIQRSKHABIPRH
|
6.8 | IC50 | 15 | — | |
OWRXHGAFWZFFCW
|
6.8 | Ki | 113 | — | |
UVBKNBPCVRBUTF
|
6.8 | IC50 | 5 | — | |
LAUHLGUSVSJYCI
|
6.8 | IC50 | 16 | — | |
NZIQNLGMMJGSQU
|
6.8 | IC50 | 6 | — | |
LUJZZYWHBDHDQX
|
6.7 | IC50 | 3 | — | |
FLEAYYMORDPWAJ
|
6.7 | Ki | 90 | — | |
HEKAIDKUDLCBRU
|
6.7 | Ki | 20 | — | |
NGRPMJQQEJIEMF
|
6.7 | IC50 | 3 | — | |
UDVRGRBOAMOTGS
|
6.7 | IC50 | 4 | — | |
WPHKIQPVPYJNAX
|
6.7 | Ki | 81 | — | |
ZVPDNRVYHLRXLX
|
6.7 | Ki | 35 | Yes | |
HCONVOOBXMEDII
|
6.7 | IC50 | 4 | — | |
VWCZORWQNKCYGE
|
6.7 | IC50 | 17 | — | |
PEGQWGLLBPWDAS
|
6.7 | IC50 | 4 | — | |
AAKJLRGGTJKAMG
|
6.6 | IC50 | 50 | Yes | |
JBGMOEFHUIKRFN
|
6.6 | IC50 | 3 | — | |
TURWKCNNQKWOTA
|
6.6 | IC50 | 3 | Yes | |
VTJHGMZHVOXJPG
|
6.6 | IC50 | 15 | — | |
WTCWMZHEAXFWPJ
|
6.6 | IC50 | 4 | — | |
XFXOYVZSTQCSQN
|
6.6 | IC50 | 3 | — | |
GFZZUAFZBKEOHV
|
6.6 | IC50 | 7 | — | |
QHUDPFOODLMGQO
|
6.6 | IC50 | 5 | — | |
KWBKHNYGQSAYCE
|
6.6 | IC50 | 3 | — |