Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HNVQCOJZTIBBPB
|
7.4 | IC50 | 3 | — | |
JFBQFAKGLQJGIL
|
7.4 | IC50 | 3 | — | |
LZECOFRPCLZCOI
|
7.4 | IC50 | 4 | — | |
QZMGOBDHHJBODW
|
7.4 | IC50 | 4 | — | |
YMSXHRWUGLAAKL
|
7.4 | IC50 | 14 | Yes | |
QYBXJSPKRPAHQB
|
7.3 | IC50 | 3 | — | |
VSFINVOSLLRTIP
|
7.3 | IC50 | 6 | — | |
LSPANGZZENHZNJ
|
7.3 | IC50 | 10 | Yes | |
ZYVUNNQGVXTJSW
|
7.3 | IC50 | 4 | — | |
FCVXPCQHDKWFDB
|
7.3 | IC50 | 3 | — | |
QFMCOTDYFYKZNH
|
7.3 | IC50 | 4 | — | |
TVJRDCQUZMGBAB
|
7.3 | IC50 | 13 | — | |
YXOXHAUUTIOBDA
|
7.3 | IC50 | 3 | Yes | |
ZMNWFTYYYCSSTF
|
7.3 | Ki | 18 | — | |
RKUBYGFDHATQAZ
|
7.3 | IC50 | 4 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 13 | — | |
BCFGMOOMADDAQU
|
7.3 | IC50 | 6 | Yes | |
PAFOOYBINUNMGT
|
7.3 | IC50 | 6 | Yes | |
ZBNZXTGUTAYRHI
|
7.3 | Kd | 102 | Yes | |
JFCHPYHJJFGZSB
|
7.2 | IC50 | 3 | Yes | |
LSJWYMSFUWBGPN
|
7.2 | IC50 | 17 | — | |
CJIJVEOGUOJOMJ
|
7.2 | IC50 | 3 | — | |
XWHJPZMQYNMSOJ
|
7.2 | IC50 | 4 | — | |
IYNUCTYYDUIRAG
|
7.2 | IC50 | 3 | — | |
RRXVMGHOCPACNG
|
7.2 | IC50 | 6 | Yes | |
IEZFFFOOLULQBR
|
7.2 | IC50 | 4 | — | |
JUSWPUDQOKINJO
|
7.2 | IC50 | 16 | — | |
UQILHDPEYNQZHG
|
7.2 | IC50 | 2 | — | |
FNYHTKUCTLSINN
|
7.2 | IC50 | 3 | Yes | |
RBBZLSVNHVBMRU
|
7.2 | IC50 | 3 | — | |
FAFWJMNGAWQHOH
|
7.2 | IC50 | 5 | — | |
WFWGCFGIGNLAGO
|
7.2 | IC50 | 4 | — | |
OPHSZSZDICRBPP
|
7.2 | IC50 | 16 | — | |
GHQPLJWMCNPRIH
|
7.1 | IC50 | 3 | Yes | |
HMXWMMRCKSDFCV
|
7.1 | IC50 | 10 | Yes | |
LVXJQMNHJWSHET
|
7.1 | IC50 | 7 | — | |
GZYUJXFTHLKPAK
|
7.1 | IC50 | 16 | — | |
GFMMDHSSOIPFTF
|
7.1 | IC50 | 2 | — | |
IQOJCGLNXTVHOS
|
7.1 | IC50 | 2 | — | |
AVHNHPHSQMBYAJ
|
7.1 | IC50 | 3 | — | |
UYJNQQDJUOUFQJ
|
7.1 | Ki | 68 | — | |
XYFZVVYVIFJBIS
|
7.1 | IC50 | 17 | — | |
QMOJTBYMFQXLLU
|
7.1 | IC50 | 6 | Yes | |
LJRGBEPLXWZRBM
|
7.1 | IC50 | 3 | — | |
JGLZFCYSDWVBJK
|
7.0 | IC50 | 2 | — | |
NBXCNCMWLZADMG
|
7.0 | IC50 | 2 | — | |
ZFDGMDVYMNWICG
|
7.0 | IC50 | 10 | — | |
YLFINAUVWATNCS
|
7.0 | IC50 | 3 | — | |
HKJUUPKKOAGVDB
|
7.0 | IC50 | 6 | Yes | |
MWFMVXZUTVIRRN
|
7.0 | IC50 | 2 | — |