Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWCCWSWQAFETLG
|
7.9 | IC50 | 4 | — | |
GFPQRHXCPZSHRH
|
7.9 | IC50 | 3 | — | |
OMYOVWAUIIJSPG
|
7.9 | IC50 | 3 | Yes | |
CMMUJJHJYMYOJR
|
7.8 | IC50 | 4 | — | |
KABLMFMHWJFKIW
|
7.8 | IC50 | 2 | — | |
LOFBARGGJCBDJT
|
7.8 | IC50 | 4 | — | |
CVBABGVEYUMHNU
|
7.8 | IC50 | 6 | — | |
PKKRQPPSMXAKFM
|
7.8 | IC50 | 3 | Yes | |
VYZQSAKXLMEDCB
|
7.8 | IC50 | 9 | — | |
WDENQIQQYWYTPO
|
7.8 | IC50 | 8 | — | |
WZZXMNBOPNKKSX
|
7.8 | Ki | 10 | — | |
SJMHQTPAHZSCGB
|
7.8 | IC50 | 4 | — | |
XKZQZMSAWVDRSP
|
7.8 | IC50 | 39 | Yes | |
ATULKYAWEUGYSF
|
7.7 | IC50 | 3 | — | |
GKFYUJHVBXYBEI
|
7.7 | IC50 | 4 | — | |
JEXCBQDTESMXHL
|
7.7 | IC50 | 3 | — | |
DYYZXRCFCVDSKD
|
7.7 | IC50 | 3 | Yes | |
HHAXMCRVXIYOJR
|
7.7 | IC50 | 4 | — | |
VVIRSVARIBXZHS
|
7.7 | IC50 | 4 | — | |
ABLXXKUDDSMAHU
|
7.7 | IC50 | 4 | — | |
KZMQPYCXSAGLTB
|
7.7 | IC50 | 8 | — | |
YOLVGSGGIWJSLQ
|
7.7 | IC50 | 3 | — | |
FUZSHLVNKZZEKR
|
7.6 | IC50 | 16 | — | |
MJLGATKKRYTQPD
|
7.6 | IC50 | 3 | — | |
SRSQULBCTWSVKL
|
7.6 | IC50 | 15 | — | |
UBPYILGKFZZVDX
|
7.6 | Kd | 130 | Yes | |
AILRADAXUVEEIR
|
7.6 | IC50 | 75 | — | |
AYIGALYNJFDMRN
|
7.6 | IC50 | 4 | — | |
RWQIOAPAHWFTMQ
|
7.6 | IC50 | 4 | — | |
SLSKTJBHIGULOP
|
7.6 | IC50 | 3 | — | |
GCUYIMVZVRRUPD
|
7.5 | IC50 | 3 | — | |
ITTRLTNMFYIYPA
|
7.5 | Kd | 17 | — | |
PQMINPFSUDRKEW
|
7.5 | IC50 | 3 | — | |
JFEKMLAOHVYFGS
|
7.5 | IC50 | 4 | — | |
DLQXAWIVHRHOQT
|
7.5 | IC50 | 6 | Yes | |
MHJBSGVISQZKDI
|
7.5 | IC50 | 4 | — | |
CDISOBGWDHAHGF
|
7.5 | IC50 | 16 | — | |
FLFHZVYTVPANLR
|
7.5 | IC50 | 4 | — | |
BWWLZGAQCJRAGF
|
7.5 | IC50 | 4 | — | |
OXAZPVDJCIJPFP
|
7.5 | IC50 | 4 | — | |
OPKHZFMFWCMAPS
|
7.4 | IC50 | 6 | — | |
SKBWQUPLWQUWPH
|
7.4 | IC50 | 6 | Yes | |
WDQXCAKHPJSZET
|
7.4 | IC50 | 3 | — | |
GAYUJMWHGBAPKD
|
7.4 | IC50 | 3 | — | |
MCEJMTKEBSFUJK
|
7.4 | IC50 | 4 | — | |
QUIWHXQETADMGN
|
7.4 | IC50 | 4 | — | |
FPGRQRNSVWYTAO
|
7.4 | IC50 | 2 | — | |
YROLHQZDEFQCCR
|
7.4 | IC50 | 4 | — | |
CZRDEUGQKBEMMH
|
7.4 | IC50 | 3 | — | |
NNGVMERLTTVLQP
|
7.4 | IC50 | 8 | — |