Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KIMIFWRATWXZEO
|
8.4 | IC50 | 3 | — | |
NYCRPERPKUAEHF
|
8.4 | IC50 | 3 | — | |
PRTPANUTPYMUDM
|
8.4 | IC50 | 3 | — | |
RSEKNDZBPQNPGL
|
8.4 | IC50 | 3 | — | |
UWXSAYUXVSFDBQ
|
8.4 | IC50 | 6 | — | |
WJGBEIOIHHBCIV
|
8.4 | IC50 | 3 | — | |
OETCDAITXCDXIB
|
8.4 | IC50 | 3 | Yes | |
JZSLVCXMHPNGNA
|
8.3 | IC50 | 5 | — | |
CRSYKTDYLTZPGM
|
8.3 | IC50 | 3 | — | |
AEBKFOMFJMJUFH
|
8.3 | IC50 | 3 | — | |
BFSRTTWIPACGMI
|
8.3 | IC50 | 4 | — | |
GNIFAULXFNJRKN
|
8.3 | IC50 | 4 | — | |
NFMGZVPRGVERNN
|
8.3 | Ki | 44 | — | |
PWLHYVUELGJGPD
|
8.3 | IC50 | 3 | — | |
UMBIRSZUCJNBHB
|
8.3 | IC50 | 18 | — | |
GCDSDVNITVBCDW
|
8.3 | IC50 | 17 | — | |
BTWVWABAWDKQNJ
|
8.3 | IC50 | 8 | — | |
HNFWPMOZPVUYBB
|
8.2 | IC50 | 4 | — | |
ACNYXAIBELJFSP
|
8.2 | IC50 | 3 | — | |
WPKVIBFJECQBCV
|
8.2 | IC50 | 3 | — | |
QTRVZMFRXOALDJ
|
8.2 | IC50 | 3 | Yes | |
QXIOZIFTPMAING
|
8.2 | IC50 | 17 | — | |
ULXXDDBFHOBEHA
|
8.2 | IC50 | 15 | Yes | |
PZWSKESWDIFAFK
|
8.2 | IC50 | 9 | — | |
PEOYVSCYYMEJBB
|
8.2 | IC50 | 3 | Yes | |
YBEIPHUFRFGXCJ
|
8.2 | IC50 | 4 | — | |
TVQHGTHLBVLBIA
|
8.1 | IC50 | 3 | Yes | |
VEQYCEHJTJSHLO
|
8.1 | IC50 | 4 | — | |
QWAHCSOEUYGXDS
|
8.1 | IC50 | 4 | — | |
FDVSOQRNTAPCHB
|
8.1 | Ki | 40 | — | |
IWDBZVDOUJFIND
|
8.1 | IC50 | 5 | — | |
FGYHOZIXSUEJDM
|
8.1 | IC50 | 3 | — | |
SCSKESFIGNPXKD
|
8.1 | IC50 | 4 | — | |
UVWRRZRGHPHHLL
|
8.1 | IC50 | 4 | — | |
SVLLKLFGGWAXTK
|
8.1 | IC50 | 5 | — | |
FXRLTQRMUHOCQN
|
8.0 | IC50 | 4 | — | |
YYNUBPUXFJKWOK
|
8.0 | IC50 | 4 | — | |
GOOMNGHXGYAHJM
|
8.0 | IC50 | 7 | — | |
KJUCPVIVNLPLEE
|
8.0 | IC50 | 10 | — | |
KPSPYNLYPZNCGV
|
8.0 | IC50 | 3 | — | |
LZOXKAMRMJSFJT
|
8.0 | IC50 | 3 | — | |
OMZCMEYTWSXEPZ
|
8.0 | IC50 | 43 | Yes | |
SRUYMJRFVGLQDV
|
8.0 | Ki | 37 | — | |
VHGQJLWYOGRRAE
|
8.0 | IC50 | 4 | — | |
IZRQFKYNXNFFQT
|
8.0 | IC50 | 3 | — | |
JXDYOSVKVSQGJM
|
8.0 | IC50 | 7 | — | |
LCFFREMLXLZNHE
|
8.0 | IC50 | 2 | — | |
UMWZSZYWDMVROC
|
8.0 | IC50 | 3 | Yes | |
BTYYWOYVBXILOJ
|
7.9 | IC50 | 4 | Yes | |
HTUBKQUPEREOGA
|
7.9 | IC50 | 6 | Yes |