Target Details
| UniProt AC | Q15303 |
|---|---|
| Gene Symbol | ERBB4 |
| Protein Name | Receptor tyrosine-protein kinase erbB-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF14843 (GF_recep_IV) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) PF21314 (TM_ErbB1) |
Summary
- Multi-target molecules 336
- Clinical molecules 58
- Avg pChEMBL 7.33
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCYSSHSIKSARGO
|
10.0 | IC50 | 19 | — | |
DLPSDPPZXRJQOY
|
9.3 | IC50 | 3 | Yes | |
KJRVCMVPIKELBC
|
9.2 | IC50 | 12 | — | |
GYFAPMADUQCILZ
|
9.2 | IC50 | 5 | — | |
MVZGYPSXNDCANY
|
9.1 | IC50 | 3 | — | |
PXBVPDIMCOILPS
|
9.1 | IC50 | 3 | Yes | |
FOOPCYOJMREECW
|
9.1 | IC50 | 5 | — | |
CNRMVFRKCDVXKW
|
9.0 | IC50 | 3 | — | |
DPNQFVJNRXPIOB
|
9.0 | IC50 | 3 | — | |
JJHXVSSJRMTBMC
|
9.0 | IC50 | 3 | Yes | |
VIANWBJPMVJZPN
|
8.9 | IC50 | 3 | Yes | |
YAPFODKXVWEFPW
|
8.9 | IC50 | 3 | — | |
ZAWWCTXYZTURLN
|
8.9 | IC50 | 4 | — | |
JGSKJUYVTDKFKT
|
8.8 | IC50 | 3 | — | |
ATUXFPJRTSKHFB
|
8.8 | IC50 | 3 | — | |
RNOAOAWBMHREKO
|
8.8 | IC50 | 15 | — | |
IMLBZWHQWRDARS
|
8.8 | IC50 | 4 | — | |
JFUDQORFBVGLMB
|
8.8 | IC50 | 3 | — | |
RHNCTEJANSMRNV
|
8.8 | IC50 | 3 | Yes | |
FKXXCQSSSCJHOZ
|
8.7 | IC50 | 3 | Yes | |
KJBZQIKLKWQVLL
|
8.7 | IC50 | 3 | — | |
KCHHPNMKOHRFDK
|
8.7 | IC50 | 3 | — | |
OMVRJIWYIOEXTO
|
8.7 | IC50 | 3 | — | |
OONFNUWBHFSNBT
|
8.7 | IC50 | 11 | — | |
WTWFBKFNVCFROY
|
8.7 | IC50 | 3 | — | |
ISEHGRGNSOYPTL
|
8.6 | IC50 | 3 | Yes | |
JWNPDZNEKVCWMY
|
8.6 | Kd | 57 | Yes | |
ROHJEIACUNTGFP
|
8.6 | IC50 | 16 | — | |
XYFPWWZEPKGCCK
|
8.6 | IC50 | 34 | — | |
AUMBQDJVOLYTCC
|
8.5 | IC50 | 3 | — | |
GDRLJBDXWDATLA
|
8.5 | IC50 | 13 | — | |
HNYGKXWZBOTZFA
|
8.5 | IC50 | 3 | — | |
KZVDSZYFRUKCEQ
|
8.5 | IC50 | 3 | — | |
NELOELKXGMSYHF
|
8.5 | IC50 | 3 | — | |
NWZQTNDYDHXMOE
|
8.5 | IC50 | 3 | — | |
OCPAAPUDKSPSJT
|
8.5 | IC50 | 3 | — | |
UCBARNSJTRWXQT
|
8.5 | IC50 | 3 | — | |
UVWRRZRGHPHHLL
|
8.5 | IC50 | 3 | — | |
RVCKMZIQUFKZFD
|
8.5 | IC50 | 7 | — | |
SSDFTYWIYVWCIE
|
8.5 | IC50 | 17 | — | |
AZSRSNUQCUDCGG
|
8.5 | IC50 | 4 | — | |
SMOPKEHQPPXRSH
|
8.5 | IC50 | 8 | — | |
UAXLMFNKXDVZKH
|
8.5 | IC50 | 3 | — | |
KTOOFDBYBSZFDL
|
8.4 | IC50 | 3 | — | |
AQEJOYTVPDGMEW
|
8.4 | IC50 | 3 | — | |
ASXBFKMZPZRWDW
|
8.4 | IC50 | 3 | — | |
BIHYRPIDCXHQKD
|
8.4 | IC50 | 3 | — | |
CQZRHVILVDPGCV
|
8.4 | IC50 | 3 | — | |
JABKEJXCSLSSEV
|
8.4 | IC50 | 3 | — | |
JLWZRGNJHZVVKD
|
8.4 | IC50 | 3 | — |