Target Details
| UniProt AC | Q15139 |
|---|---|
| Gene Symbol | PRKD1 |
| Protein Name | Serine/threonine-protein kinase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 208
- Clinical molecules 105
- Avg pChEMBL 7.25
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (208)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
YBYYWUUUGCNAHQ
|
6.5 | IC50 | 8 | — | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
XQVVPGYIWAGRNI
|
6.5 | Kd | 34 | — | |
OBRQLJITIRIMLQ
|
6.5 | IC50 | 11 | — | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
HZCVZGCAUBUBST
|
6.5 | IC50 | 3 | — | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | IC50 | 147 | Yes | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
HHLKZSJXDAZIGG
|
6.4 | IC50 | 10 | Yes | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
SNQKPKFVSANKFP
|
6.3 | IC50 | 6 | — | |
SSNQAUBBJYCSMY
|
6.3 | IC50 | 5 | — | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 82 | Yes | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
HDAJDNHIBCDLQF
|
6.3 | IC50 | 14 | — | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
QQKKPWJFHBFCTH
|
6.2 | IC50 | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.2 | Ki | 10 | Yes | |
ZUKHVOLIPVGCHQ
|
6.2 | Ki | 10 | Yes | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
CJTQBCMGMLTHPI
|
6.2 | IC50 | 4 | — | |
HZTYDQRUAWIZRE
|
6.2 | Kd | 40 | Yes | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
WZOQKGRFRIFIEB
|
6.1 | IC50 | 3 | — | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
JWNPDZNEKVCWMY
|
6.1 | Kd | 57 | Yes | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
XSHQBIXMLULFEV
|
6.0 | IC50 | 13 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |