Target Details
| UniProt AC | Q15139 |
|---|---|
| Gene Symbol | PRKD1 |
| Protein Name | Serine/threonine-protein kinase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 208
- Clinical molecules 105
- Avg pChEMBL 7.25
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (208)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OFPFIAWWDTYSBZ
|
7.1 | Ki | 15 | Yes | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
RHLRPKGACJKWPF
|
7.1 | IC50 | 12 | Yes | |
GGQAEINRBKFRGZ
|
7.1 | IC50 | 15 | Yes | |
KGMSYXGSYGEHIS
|
7.1 | IC50 | 4 | — | |
NHDDTLMPCVOXFH
|
7.1 | IC50 | 16 | Yes | |
SXDPQGRNHSLZPC
|
7.0 | IC50 | 18 | — | |
MQCCJEYZKWZQHU
|
7.0 | IC50 | 15 | Yes | |
YSVVBGPTTSJYPA
|
7.0 | IC50 | 13 | Yes | |
PFAZIMNYEBJHOA
|
7.0 | IC50 | 12 | Yes | |
XRFOMFNAMTYCFF
|
7.0 | IC50 | 12 | Yes | |
YUAWUNMKPARPJD
|
7.0 | IC50 | 14 | Yes | |
BERLXWPRSBJFHO
|
7.0 | IC50 | 4 | — | |
RBZLXANOQRQGTN
|
7.0 | IC50 | 3 | — | |
ZUYALLZMSFUHFE
|
7.0 | IC50 | 3 | — | |
FWXIKQAZCDAIKV
|
6.9 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
6.9 | IC50 | 15 | Yes | |
FTCSRLCKGZJDCK
|
6.9 | IC50 | 3 | — | |
OGJTZCZJWZSZBT
|
6.9 | IC50 | 12 | Yes | |
VWHZWDRIMLETBG
|
6.9 | IC50 | 12 | Yes | |
DRCBMJUPXHWGMN
|
6.8 | IC50 | 15 | Yes | |
JWVXPOMGWPAEAJ
|
6.8 | IC50 | 10 | Yes | |
QNULKTUETCUJKC
|
6.8 | IC50 | 14 | Yes | |
CZIVUSJISIAXJB
|
6.8 | IC50 | 18 | — | |
OOPMDKIRVTXOPT
|
6.8 | IC50 | 11 | — | |
JCHWETQOLSPUBV
|
6.8 | IC50 | 14 | — | |
JHKZENPNLYAVCT
|
6.8 | IC50 | 15 | Yes | |
OQSTWXKHTZWKLD
|
6.8 | IC50 | 15 | Yes | |
AACFPJSJOWQNBN
|
6.7 | IC50 | 4 | — | |
AWJAAKKEYXUCFY
|
6.7 | IC50 | 5 | — | |
DQYBRTASHMYDJG
|
6.7 | IC50 | 13 | Yes | |
LGSHHKIOBFPSEK
|
6.7 | IC50 | 12 | Yes | |
AILRADAXUVEEIR
|
6.7 | IC50 | 75 | — | |
GGFLGGNNYKCRAV
|
6.7 | IC50 | 3 | — | |
BOJKFRKNLSCGHY
|
6.7 | Ki | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.7 | Ki | 10 | Yes | |
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
GAEKZIARZJRZTM
|
6.7 | IC50 | 3 | — | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
GDQXJQSQYMMKRA
|
6.6 | IC50 | 15 | — | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
QMGUOJYZJKLOLH
|
6.6 | IC50 | 21 | Yes | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes |