Target Details
| UniProt AC | Q15139 |
|---|---|
| Gene Symbol | PRKD1 |
| Protein Name | Serine/threonine-protein kinase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 208
- Clinical molecules 105
- Avg pChEMBL 7.25
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (208)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WMFOYAZROOMVDL
|
7.8 | IC50 | 3 | — | |
CXSQMXRQOZZFLD
|
7.8 | IC50 | 18 | — | |
NPHRPHMHAOPRTH
|
7.8 | IC50 | 2 | — | |
PBCZSGKMGDDXIJ
|
7.8 | IC50 | 68 | Yes | |
SCJXQZZYGYLKJG
|
7.8 | IC50 | 3 | — | |
VAVGLCQDZFLPHS
|
7.8 | IC50 | 3 | — | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
VJHWVSYYFZRUEK
|
7.7 | IC50 | 3 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
CNLCKMDXRXVYMV
|
7.7 | IC50 | 3 | — | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
AYCPARAPKDAOEN
|
7.7 | IC50 | 73 | — | |
GMFDXTZCWCUHOB
|
7.6 | Ki | 2 | — | |
NVHXHWFKRHCFCI
|
7.6 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
DHUAGGSHTKPOHU
|
7.5 | IC50 | 3 | — | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
KOZFSFOOLUUIGY
|
7.5 | IC50 | 88 | Yes | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
GTWNYADDKACXSW
|
7.5 | IC50 | 3 | — | |
ZACCEWDQLIBKAZ
|
7.5 | IC50 | 2 | — | |
ZHMXXVNQAFCXKK
|
7.5 | IC50 | 15 | — | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
PNZJIQBIMCZAKU
|
7.3 | IC50 | 3 | — | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
BMGQWWVMWDBQGC
|
7.3 | IC50 | 91 | Yes | |
CEWOYNHYISZPFC
|
7.3 | IC50 | 3 | — | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
LTWPQYSXDJCNBR
|
7.3 | IC50 | 3 | — | |
GVSRILDMSGVJTR
|
7.2 | IC50 | 7 | — | |
HZWIAHGTTPPVAC
|
7.2 | Ki | 2 | — | |
VWVYILCFSYNJHF
|
7.2 | IC50 | 49 | — | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes | |
FZJMLWNUSUKYPU
|
7.2 | Ki | 2 | — | |
NRUVICOXXLOXCB
|
7.2 | IC50 | 13 | Yes | |
WHROQBPMBHWWTB
|
7.2 | IC50 | 3 | — | |
WXGCJNLWHYWDFU
|
7.2 | IC50 | 3 | — | |
MGMNDPRNDCWSMZ
|
7.2 | IC50 | 12 | Yes | |
GRENHRYHWHSBLM
|
7.1 | IC50 | 12 | Yes | |
LGCKGDRUTNACTA
|
7.1 | IC50 | 11 | — |