Target Details
| UniProt AC | Q15139 |
|---|---|
| Gene Symbol | PRKD1 |
| Protein Name | Serine/threonine-protein kinase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 208
- Clinical molecules 105
- Avg pChEMBL 7.25
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (208)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
FZJMLWNUSUKYPU
|
9.1 | Ki | 2 | — | |
HCMOZLPTNMKKAS
|
9.0 | IC50 | 3 | — | |
KKMZQQWZVBKDFC
|
9.0 | IC50 | 3 | — | |
MTXHXAFTVABHOY
|
9.0 | IC50 | 3 | — | |
NCAVLXJPDIQUIS
|
9.0 | IC50 | 3 | — | |
SCJXQZZYGYLKJG
|
9.0 | IC50 | 3 | — | |
VDRJYOAEHZMFEB
|
9.0 | IC50 | 3 | — | |
XBDRAUPLGHAFCU
|
9.0 | IC50 | 3 | — | |
XNWDRALEEPGBHB
|
9.0 | IC50 | 3 | — | |
YKWMQNUCOUUHQO
|
9.0 | IC50 | 3 | — | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
WXGCJNLWHYWDFU
|
8.7 | IC50 | 3 | — | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
HZWIAHGTTPPVAC
|
8.4 | Ki | 2 | — | |
VBWZGQKYVCFADL
|
8.4 | IC50 | 3 | — | |
ZIATUPKJNZVSLT
|
8.4 | IC50 | 3 | — | |
RODIOQSCTKCZKO
|
8.4 | Ki | 2 | — | |
DIZACSOTRSXCHC
|
8.4 | IC50 | 4 | — | |
QYHQDVASMWOBHE
|
8.3 | Ki | 2 | — | |
HXYGELZVZAPWID
|
8.3 | IC50 | 3 | — | |
XYUFCXJZFZPEJD
|
8.3 | Ki | 23 | Yes | |
LSEXYAQECWMUPY
|
8.3 | IC50 | 3 | — | |
OHSPVJFJVRIKGA
|
8.2 | Ki | 2 | — | |
BQJRUJTZSGYBEZ
|
8.2 | Kd | 13 | Yes | |
LRYNHRWGDADZKP
|
8.2 | IC50 | 3 | — | |
SFSGIDJMRRLJFG
|
8.2 | IC50 | 3 | — | |
SAYMBMAHSBYKKR
|
8.2 | IC50 | 12 | Yes | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
SFSGIDJMRRLJFG
|
8.1 | IC50 | 3 | — | |
ZVKJUDYDWABBFR
|
8.1 | IC50 | 3 | — | |
POTTVLREWUNNRO
|
8.1 | IC50 | 17 | Yes | |
CDXNZQYZADSNCP
|
8.0 | IC50 | 12 | Yes | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
FFKRSNGYONHGEV
|
8.0 | IC50 | 12 | Yes | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
OPQUGNXQOSDRMT
|
8.0 | IC50 | 12 | Yes | |
PGWBJRRPIUVOAD
|
8.0 | IC50 | 12 | Yes | |
PBCZSGKMGDDXIJ
|
7.9 | IC50 | 14 | Yes | |
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
SMZYTCQRZVNFFJ
|
7.8 | IC50 | 16 | Yes | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes |