Target Details
| UniProt AC | Q15120 |
|---|---|
| Gene Symbol | PDK3 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 362
- Clinical molecules 0
- Avg pChEMBL 6.83
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (362)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JQHNJRAABZZPFN
|
6.0 | IC50 | 4 | — | |
JXGCDBJFNMMLNB
|
6.0 | IC50 | 4 | — | |
JZKWCVYCWBMBFY
|
6.0 | IC50 | 4 | — | |
JZQRWFCPYXTEEC
|
6.0 | IC50 | 4 | — | |
KHTIYNJMMLQJRX
|
6.0 | IC50 | 4 | — | |
KHWHZLYCFONFBB
|
6.0 | IC50 | 4 | — | |
KMWHNYZBANTQFA
|
6.0 | IC50 | 4 | — | |
KZGYMLHJMGQXOM
|
6.0 | IC50 | 4 | — | |
LBPOGQUABVQXPM
|
6.0 | IC50 | 4 | — | |
LMKXJIKIUSIWSP
|
6.0 | IC50 | 4 | — | |
LNBYJUPTVFIGQB
|
6.0 | IC50 | 4 | — | |
LSBCJXWWDZEWRF
|
6.0 | IC50 | 4 | — | |
LVNJKOIEYNEOMZ
|
6.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
6.0 | IC50 | 4 | — | |
MMIWOBFOVOZMKG
|
6.0 | IC50 | 4 | — | |
MMLLULKUDKWCNR
|
6.0 | IC50 | 4 | — | |
MTLYSRUJNCWFOX
|
6.0 | IC50 | 4 | — | |
NEXLZTATSAIBTR
|
6.0 | IC50 | 4 | — | |
NPZRDYRAAKIHPY
|
6.0 | IC50 | 4 | — | |
OINIDTBTTIYZIO
|
6.0 | IC50 | 4 | — | |
PABSUYDXHABXPY
|
6.0 | IC50 | 4 | — | |
PAVCFPGEDQLOLY
|
6.0 | IC50 | 4 | — | |
PUHWWAJTHDKCGR
|
6.0 | IC50 | 4 | — | |
PWDYOVIZDCYFRZ
|
6.0 | IC50 | 4 | — | |
PXUOKRBBSRTUNE
|
6.0 | IC50 | 4 | — | |
PZPMTBAIXNMBME
|
6.0 | IC50 | 4 | — | |
QMXIGKOHRUDNMV
|
6.0 | IC50 | 4 | — | |
QPFCZCMRUOQZRG
|
6.0 | IC50 | 4 | — | |
QQMKDSHSGYQMOV
|
6.0 | IC50 | 4 | — | |
QTZREWXFIMJBHN
|
6.0 | IC50 | 4 | — | |
QXCUSMAHYXWCOF
|
6.0 | IC50 | 4 | — | |
RECOPQDOXFPBNE
|
6.0 | IC50 | 4 | — | |
RFGOESLFDUAMGB
|
6.0 | IC50 | 4 | — | |
RTVPWYJBMHEYTA
|
6.0 | IC50 | 4 | — | |
RWEVXAYNUMFKQD
|
6.0 | IC50 | 4 | — | |
SLUNFEBZDXASNJ
|
6.0 | IC50 | 4 | — | |
SVXHTPKAAXLDLX
|
6.0 | IC50 | 4 | — | |
SYPAMOJTLDNMQL
|
6.0 | IC50 | 4 | — | |
UDUFRUMXLFCNQN
|
6.0 | IC50 | 4 | — | |
UKVBAJDPXOGHTO
|
6.0 | IC50 | 4 | — | |
UUGBZZQAHRXVBV
|
6.0 | IC50 | 4 | — | |
UZZOOCJSVGDZPS
|
6.0 | IC50 | 4 | — | |
VAEZIOUPBWPWKT
|
6.0 | IC50 | 4 | — | |
VKRJGZNMDIROFE
|
6.0 | IC50 | 4 | — | |
VLHPKUJISXSNFG
|
6.0 | IC50 | 4 | — | |
WHGYCNIXXDEKMI
|
6.0 | IC50 | 4 | — | |
WILCKYMTSIVKIZ
|
6.0 | IC50 | 4 | — | |
WLNHFWZZOOBEHX
|
6.0 | IC50 | 4 | — | |
WLSKWMBVRHXLLG
|
6.0 | IC50 | 4 | — | |
WREUMGOBADOOMR
|
6.0 | IC50 | 4 | — |