Target Details
| UniProt AC | Q15120 |
|---|---|
| Gene Symbol | PDK3 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 362
- Clinical molecules 0
- Avg pChEMBL 6.83
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (362)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XVLUOKHYAJARDM
|
7.0 | IC50 | 4 | — | |
YDTBZYAJXNXQGG
|
7.0 | IC50 | 4 | — | |
YKCSCWCEGAZILJ
|
7.0 | IC50 | 4 | — | |
YQIDANKABBOUGC
|
7.0 | IC50 | 4 | — | |
YTDJEAZYTGIAJJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — | |
ZPMRFYJDPARNBL
|
7.0 | IC50 | 4 | — | |
ZUZGRFYAGRDPGJ
|
7.0 | IC50 | 4 | — | |
ZVFIHSAIQWKOAE
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZYAAUDLDGUEAPN
|
7.0 | IC50 | 4 | — | |
ZYLSRWYAGYUONP
|
7.0 | IC50 | 4 | — | |
CJKPVNLQNOSPAE
|
7.0 | IC50 | 4 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
URBQRLTYIDBJQO
|
7.0 | IC50 | 4 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
DTDZLJHKVNTQGZ
|
6.9 | IC50 | 4 | — | |
MWKSRKSEWLRPBL
|
6.9 | Kd | 1075 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
KOAXITXTHITWLT
|
6.9 | IC50 | 4 | — | |
NSEKNXMDWSTZJL
|
6.9 | IC50 | 4 | — | |
XNGVNSXRRADPSC
|
6.9 | IC50 | 4 | — | |
TYTXGPAMIGYEGN
|
6.9 | IC50 | 4 | — | |
TWRWVLYTPAORIW
|
6.8 | IC50 | 4 | — | |
VPETUWRKODTKNY
|
6.8 | IC50 | 4 | — | |
YWAFKNHDMNEFPA
|
6.8 | IC50 | 2 | — | |
CWHNQKPCYFFKDR
|
6.8 | IC50 | 4 | — | |
ZOPYDEDEHVUGTC
|
6.8 | IC50 | 4 | — | |
LDFLSIZNFQLCDQ
|
6.8 | IC50 | 4 | — | |
GFICNEUSPWSTPP
|
6.8 | IC50 | 4 | — | |
OXQTXJIDMWRZLX
|
6.7 | IC50 | 4 | — | |
SFQMDVJNIAAAJA
|
6.7 | IC50 | 4 | — | |
HVZAUSYZLGXKIP
|
6.7 | IC50 | 4 | — | |
QRPZFMFZNJHOTN
|
6.6 | IC50 | 4 | — | |
GAFYAXXDUJHTEI
|
6.6 | IC50 | 4 | — | |
RTYCQDBBCMTUFF
|
6.6 | IC50 | 4 | — | |
XJVOPOWBIDUKFI
|
6.5 | IC50 | 4 | — | |
ZTSYVKWXYINLJV
|
6.5 | IC50 | 4 | — | |
AUJRIOZTXXHUGR
|
6.5 | IC50 | 4 | — | |
BQRFDZQRKCARHX
|
6.5 | IC50 | 4 | — | |
BTVCELJQYVYBMY
|
6.5 | IC50 | 4 | — | |
DXULLUCLDXLAEE
|
6.5 | IC50 | 4 | — | |
KCXGMKDIPWGLSK
|
6.5 | IC50 | 4 | — | |
KURLHYDERFSDAV
|
6.5 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
6.5 | IC50 | 4 | — |