Target Details
| UniProt AC | Q15120 |
|---|---|
| Gene Symbol | PDK3 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 362
- Clinical molecules 0
- Avg pChEMBL 6.83
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (362)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBLPPJHSHGACEJ
|
7.0 | IC50 | 4 | — | |
FHANGEZWICYMAN
|
7.0 | IC50 | 4 | — | |
FHCJWURPGGJVIU
|
7.0 | IC50 | 4 | — | |
FLMXFYUZYPWMHO
|
7.0 | IC50 | 4 | — | |
FPKYIUHRFOETKG
|
7.0 | IC50 | 4 | — | |
FUJJLTFFZUJRAF
|
7.0 | IC50 | 4 | — | |
FURRPKJZBWBALL
|
7.0 | IC50 | 4 | — | |
FVWCFDQTLRXQFX
|
7.0 | IC50 | 4 | — | |
GAEIKTXZNLANQY
|
7.0 | IC50 | 4 | — | |
GIFBFVKPOAPOQF
|
7.0 | IC50 | 4 | — | |
GOYZFCBIPVDHLA
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
HBQAMWIICPEKLM
|
7.0 | IC50 | 4 | — | |
HEZXCHOQRVOWOO
|
7.0 | IC50 | 4 | — | |
HMDVVVVFTDRVEN
|
7.0 | IC50 | 4 | — | |
HOTHCUMDFKWXAY
|
7.0 | IC50 | 4 | — | |
HPKSWZBPOBFFGH
|
7.0 | IC50 | 4 | — | |
HQXGHFGYLLOUQN
|
7.0 | IC50 | 4 | — | |
HUZNUFRXRYRKLQ
|
7.0 | IC50 | 4 | — | |
HXGAMFVEHXJPPA
|
7.0 | IC50 | 4 | — | |
IAOKECPRCAJJLW
|
7.0 | IC50 | 4 | — | |
IBOAFKTZBFJUKA
|
7.0 | IC50 | 4 | — | |
IJYGCXRXUFNBBX
|
7.0 | IC50 | 4 | — | |
IRGFJNBJMFGIAK
|
7.0 | IC50 | 4 | — | |
JEULTWLFDMZUPQ
|
7.0 | IC50 | 4 | — | |
JITAWAABXAQPMA
|
7.0 | IC50 | 4 | — | |
JKSGRMDJMCJGOZ
|
7.0 | IC50 | 4 | — | |
JLVBJWREILIRAS
|
7.0 | IC50 | 4 | — | |
JLWPPFZGJGHSTJ
|
7.0 | IC50 | 4 | — | |
JMIVUIMGDJZLIG
|
7.0 | IC50 | 4 | — | |
JNGRLPFNEIFOTG
|
7.0 | IC50 | 4 | — | |
JOCFMBDFPBFGGL
|
7.0 | IC50 | 4 | — | |
JOJIFEAFJOWRTN
|
7.0 | IC50 | 4 | — | |
KLQHYYHEUCEROZ
|
7.0 | IC50 | 4 | — | |
KLQHYYHEUCEROZ
|
7.0 | IC50 | 4 | — | |
KUUZLDUCOUHSFK
|
7.0 | IC50 | 4 | — | |
KZUMTKNLJKJSBD
|
7.0 | IC50 | 4 | — | |
KZUMTKNLJKJSBD
|
7.0 | IC50 | 4 | — | |
LKBFKOYSSYSDQH
|
7.0 | IC50 | 4 | — | |
LLGHHTDOUJTEOP
|
7.0 | IC50 | 4 | — | |
LLWJFRPCKCAMKV
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LSEQOPAXXJYNDG
|
7.0 | IC50 | 4 | — | |
LSJRQFSUVPSXTH
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
MJDOETCLTIAWPE
|
7.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
7.0 | IC50 | 4 | — |