Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AFRYLLNYYFRUKZ
|
6.0 | IC50 | 4 | — | |
AGIRAUWGTYSFEY
|
6.0 | IC50 | 4 | — | |
AIDMBUXHQJQJMB
|
6.0 | IC50 | 4 | — | |
AVIBHWXBXPFMLQ
|
6.0 | IC50 | 4 | — | |
BOCXGAVHERNIED
|
6.0 | IC50 | 4 | — | |
BOGRKBZCGGVGGS
|
6.0 | IC50 | 4 | — | |
BVSMEZQQQTUAMN
|
6.0 | IC50 | 4 | — | |
CBHNHZXDESJXQZ
|
6.0 | IC50 | 4 | — | |
CKCBDRGQGSQRFN
|
6.0 | IC50 | 4 | — | |
CWAXXGRNESDIFD
|
6.0 | IC50 | 4 | — | |
DFBBARPBDNOHIG
|
6.0 | IC50 | 4 | — | |
DRJCGVYRZOBJOV
|
6.0 | IC50 | 4 | — | |
FBRKPMZCQHNIJI
|
6.0 | IC50 | 4 | — | |
FKHMXABMILEREF
|
6.0 | IC50 | 4 | — | |
FMLYGCPVSHVBGL
|
6.0 | IC50 | 4 | — | |
FMTIOPPCYVSTGQ
|
6.0 | IC50 | 4 | — | |
FOHLYNYTSUJQTP
|
6.0 | IC50 | 4 | — | |
FQMNWBLEFIAYPW
|
6.0 | IC50 | 4 | — | |
GHNVNCXYLHYQDO
|
6.0 | IC50 | 4 | — | |
GKSNEZLHIIZEGL
|
6.0 | IC50 | 4 | — | |
GNIVANXSNOBJOV
|
6.0 | IC50 | 4 | — | |
GXNHMFDKLVMBBF
|
6.0 | IC50 | 4 | — | |
HGWPYDZYRWUXAC
|
6.0 | IC50 | 4 | — | |
HJCYHYZYHRDVBU
|
6.0 | IC50 | 4 | — | |
HSRXRPVIBOXEKS
|
6.0 | IC50 | 4 | — | |
HXEZLTWOXMXCJJ
|
6.0 | IC50 | 4 | — | |
IEPMJKSTICKITB
|
6.0 | IC50 | 4 | — | |
JBXCZTFOQMGTBA
|
6.0 | IC50 | 4 | — | |
JCMGJBTYTUCSSM
|
6.0 | IC50 | 4 | — | |
JLWRTIPIGXDNEG
|
6.0 | IC50 | 4 | — | |
JQHAKNWHEFDSNQ
|
6.0 | IC50 | 4 | — | |
JQHNJRAABZZPFN
|
6.0 | IC50 | 4 | — | |
JXGCDBJFNMMLNB
|
6.0 | IC50 | 4 | — | |
JZKWCVYCWBMBFY
|
6.0 | IC50 | 4 | — | |
JZQRWFCPYXTEEC
|
6.0 | IC50 | 4 | — | |
KHTIYNJMMLQJRX
|
6.0 | IC50 | 4 | — | |
KHWHZLYCFONFBB
|
6.0 | IC50 | 4 | — | |
KMWHNYZBANTQFA
|
6.0 | IC50 | 4 | — | |
KZGYMLHJMGQXOM
|
6.0 | IC50 | 4 | — | |
LBPOGQUABVQXPM
|
6.0 | IC50 | 4 | — | |
LMKXJIKIUSIWSP
|
6.0 | IC50 | 4 | — | |
LNBYJUPTVFIGQB
|
6.0 | IC50 | 4 | — | |
LSBCJXWWDZEWRF
|
6.0 | IC50 | 4 | — | |
LVNJKOIEYNEOMZ
|
6.0 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
6.0 | IC50 | 4 | — | |
MMIWOBFOVOZMKG
|
6.0 | IC50 | 4 | — | |
MMLLULKUDKWCNR
|
6.0 | IC50 | 4 | — | |
MTLYSRUJNCWFOX
|
6.0 | IC50 | 4 | — | |
NEXLZTATSAIBTR
|
6.0 | IC50 | 4 | — | |
NPZRDYRAAKIHPY
|
6.0 | IC50 | 4 | — |