Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNGVNSXRRADPSC
|
6.9 | IC50 | 4 | — | |
LZCHVMYGVHFFSN
|
6.9 | IC50 | 6 | — | |
VJSMYBWGSKJUEL
|
6.9 | IC50 | 4 | — | |
CYNYZDWGNQYJDF
|
6.9 | IC50 | 3 | — | |
BTMDJLDUVYTZBI
|
6.8 | IC50 | 2 | — | |
TWRWVLYTPAORIW
|
6.8 | IC50 | 4 | — | |
VPETUWRKODTKNY
|
6.8 | IC50 | 4 | — | |
CWHNQKPCYFFKDR
|
6.8 | IC50 | 4 | — | |
TYTXGPAMIGYEGN
|
6.8 | IC50 | 4 | — | |
ZOPYDEDEHVUGTC
|
6.8 | IC50 | 4 | — | |
LDFLSIZNFQLCDQ
|
6.8 | IC50 | 4 | — | |
KKVYOWPPMNSLCP
|
6.8 | Ki | 5 | — | |
GFICNEUSPWSTPP
|
6.7 | IC50 | 4 | — | |
ZBCASIFBVICMSH
|
6.7 | IC50 | 4 | — | |
OXQTXJIDMWRZLX
|
6.7 | IC50 | 4 | — | |
MUBBTSZWDVFVLT
|
6.7 | IC50 | 3 | — | |
HVZAUSYZLGXKIP
|
6.7 | IC50 | 4 | — | |
QRPZFMFZNJHOTN
|
6.6 | IC50 | 4 | — | |
GAFYAXXDUJHTEI
|
6.6 | IC50 | 4 | — | |
RTYCQDBBCMTUFF
|
6.6 | IC50 | 4 | — | |
FLCLKDRMVXBLHR
|
6.5 | IC50 | 4 | — | |
XJVOPOWBIDUKFI
|
6.5 | IC50 | 4 | — | |
ZTSYVKWXYINLJV
|
6.5 | IC50 | 4 | — | |
AUJRIOZTXXHUGR
|
6.5 | IC50 | 4 | — | |
BQRFDZQRKCARHX
|
6.5 | IC50 | 4 | — | |
BTVCELJQYVYBMY
|
6.5 | IC50 | 4 | — | |
DXULLUCLDXLAEE
|
6.5 | IC50 | 4 | — | |
KCXGMKDIPWGLSK
|
6.5 | IC50 | 4 | — | |
KURLHYDERFSDAV
|
6.5 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
6.5 | IC50 | 4 | — | |
PYWNULWLMYXJIE
|
6.5 | IC50 | 4 | — | |
QWHBUKMSQWNPLU
|
6.5 | IC50 | 4 | — | |
REKSHMUIHDBZEL
|
6.5 | IC50 | 4 | — | |
UHLKSPFADXABBK
|
6.5 | IC50 | 4 | — | |
WQBUEPUJTZXCSW
|
6.5 | IC50 | 4 | — | |
XXFAGYMXMCJALN
|
6.5 | IC50 | 4 | — | |
XZGKZXADQIAIAB
|
6.5 | IC50 | 4 | — | |
ZPNZQVNPYMEKML
|
6.5 | IC50 | 4 | — | |
ZQLXLPNBWGVBKS
|
6.5 | IC50 | 4 | — | |
GVZALBNYLGZCKU
|
6.4 | IC50 | 2 | — | |
LHSKWVQEAJUPOG
|
6.4 | IC50 | 4 | — | |
OVUREOQFPBNHNM
|
6.4 | IC50 | 4 | — | |
VCQLZAWRWBAQKG
|
6.3 | IC50 | 2 | — | |
WRKXOYGLVREKOE
|
6.3 | IC50 | 2 | — | |
RPNZGGQCZUXPBC
|
6.2 | IC50 | 4 | — | |
JKJOXJGLLJZNII
|
6.2 | IC50 | 2 | — | |
NLHSXYGKBUOFPL
|
6.2 | IC50 | 4 | — | |
UFRHUTDVBLSOCA
|
6.2 | Ki | 2 | — | |
JAOFIBKJPAHQNQ
|
6.1 | IC50 | 4 | — | |
QGVSLEINXMWQMT
|
6.0 | IC50 | 4 | — |