Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJEXWLLUJGZGAK
|
7.0 | IC50 | 4 | — | |
SQEBZRWBDVPJDR
|
7.0 | IC50 | 4 | — | |
SWUFKVPRVHWIRW
|
7.0 | IC50 | 4 | — | |
SXBULXXRUIFERC
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
TZKXWAODTKIRQH
|
7.0 | IC50 | 4 | — | |
UDXRPQUWDSCOTK
|
7.0 | IC50 | 4 | — | |
UMRLOUSNWOYFFM
|
7.0 | IC50 | 4 | — | |
UOLOUISPBSPRGG
|
7.0 | IC50 | 4 | — | |
VIRNQTUQCWCOAV
|
7.0 | IC50 | 4 | — | |
VLTVCXJATKADNO
|
7.0 | IC50 | 4 | — | |
VPMACFXFRUVPQK
|
7.0 | IC50 | 4 | — | |
WBZWNTJAWZVNCI
|
7.0 | IC50 | 4 | — | |
WEJYENUPPGWUCM
|
7.0 | IC50 | 4 | — | |
WEWLWBDTDINJNR
|
7.0 | IC50 | 4 | — | |
WKTAYYWOLXTJGL
|
7.0 | IC50 | 4 | — | |
WQJHFNBULHHCAT
|
7.0 | IC50 | 4 | — | |
WYUKVGVZYSCCDJ
|
7.0 | IC50 | 4 | — | |
XBXCLVBYMZQBFQ
|
7.0 | IC50 | 4 | — | |
XFLXHBRVXWEPCZ
|
7.0 | IC50 | 4 | — | |
XNWFFSUKXSXYOJ
|
7.0 | IC50 | 4 | — | |
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XVLUOKHYAJARDM
|
7.0 | IC50 | 4 | — | |
YDTBZYAJXNXQGG
|
7.0 | IC50 | 4 | — | |
YKCSCWCEGAZILJ
|
7.0 | IC50 | 4 | — | |
YQIDANKABBOUGC
|
7.0 | IC50 | 4 | — | |
YTDJEAZYTGIAJJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — | |
ZPMRFYJDPARNBL
|
7.0 | IC50 | 4 | — | |
ZUZGRFYAGRDPGJ
|
7.0 | IC50 | 4 | — | |
ZVFIHSAIQWKOAE
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZYAAUDLDGUEAPN
|
7.0 | IC50 | 4 | — | |
ZYLSRWYAGYUONP
|
7.0 | IC50 | 4 | — | |
CJKPVNLQNOSPAE
|
7.0 | IC50 | 4 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
RDZHNFZDJQDIFX
|
7.0 | IC50 | 2 | — | |
URBQRLTYIDBJQO
|
7.0 | IC50 | 4 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
SFQMDVJNIAAAJA
|
7.0 | IC50 | 4 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
FUOYLHLTUNTBFV
|
6.9 | IC50 | 2 | — | |
KOAXITXTHITWLT
|
6.9 | IC50 | 4 | — | |
NSEKNXMDWSTZJL
|
6.9 | IC50 | 4 | — | |
RRFJREZCKIANGM
|
6.9 | IC50 | 2 | — |