Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADYFSAHHBUQVGK
|
7.0 | IC50 | 4 | — | |
AEROUCXDUDYEKO
|
7.0 | IC50 | 4 | — | |
APWMGNIAYJJUAF
|
7.0 | IC50 | 4 | — | |
ARUCEZREJLJFDT
|
7.0 | IC50 | 4 | — | |
BCJWSMLGFKGOGY
|
7.0 | IC50 | 4 | — | |
BEDBXCKARVIOCD
|
7.0 | IC50 | 4 | — | |
BPZOUMFIFRETCA
|
7.0 | IC50 | 4 | — | |
BQUDNQLXMYGDNQ
|
7.0 | IC50 | 4 | — | |
BSLIZBUPULPNHQ
|
7.0 | IC50 | 4 | — | |
BSLIZBUPULPNHQ
|
7.0 | IC50 | 4 | — | |
BSQGGNPQVHKELV
|
7.0 | IC50 | 4 | — | |
BYSDPXBOYDDWFZ
|
7.0 | IC50 | 4 | — | |
CAIPBEZKRVGEKE
|
7.0 | IC50 | 4 | — | |
CGIKZEQNOIDVOV
|
7.0 | IC50 | 4 | — | |
CGYZWZHPCJOISU
|
7.0 | IC50 | 4 | — | |
CGYZWZHPCJOISU
|
7.0 | IC50 | 4 | — | |
CHWXLTDPQZWFAM
|
7.0 | IC50 | 4 | — | |
CXYRJLAOPDAFSS
|
7.0 | IC50 | 4 | — | |
CXYRJLAOPDAFSS
|
7.0 | IC50 | 4 | — | |
CYESLTXMVJMIOU
|
7.0 | IC50 | 4 | — | |
DGUGNQFTCBUBEL
|
7.0 | IC50 | 4 | — | |
DTLSNWXWIAFKCH
|
7.0 | IC50 | 4 | — | |
FBLPPJHSHGACEJ
|
7.0 | IC50 | 4 | — | |
FHANGEZWICYMAN
|
7.0 | IC50 | 4 | — | |
FHCJWURPGGJVIU
|
7.0 | IC50 | 4 | — | |
FLMXFYUZYPWMHO
|
7.0 | IC50 | 4 | — | |
FPKYIUHRFOETKG
|
7.0 | IC50 | 4 | — | |
FUJJLTFFZUJRAF
|
7.0 | IC50 | 4 | — | |
FURRPKJZBWBALL
|
7.0 | IC50 | 4 | — | |
FVWCFDQTLRXQFX
|
7.0 | IC50 | 4 | — | |
GAEIKTXZNLANQY
|
7.0 | IC50 | 4 | — | |
GIFBFVKPOAPOQF
|
7.0 | IC50 | 4 | — | |
GOYZFCBIPVDHLA
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
HBQAMWIICPEKLM
|
7.0 | IC50 | 4 | — | |
HEZXCHOQRVOWOO
|
7.0 | IC50 | 4 | — | |
HMDVVVVFTDRVEN
|
7.0 | IC50 | 4 | — | |
HOTHCUMDFKWXAY
|
7.0 | IC50 | 4 | — | |
HPKSWZBPOBFFGH
|
7.0 | IC50 | 4 | — | |
HQXGHFGYLLOUQN
|
7.0 | IC50 | 4 | — | |
HUZNUFRXRYRKLQ
|
7.0 | IC50 | 4 | — | |
HXGAMFVEHXJPPA
|
7.0 | IC50 | 4 | — | |
IAOKECPRCAJJLW
|
7.0 | IC50 | 4 | — | |
IBOAFKTZBFJUKA
|
7.0 | IC50 | 4 | — | |
IJYGCXRXUFNBBX
|
7.0 | IC50 | 4 | — | |
IRGFJNBJMFGIAK
|
7.0 | IC50 | 4 | — | |
JEULTWLFDMZUPQ
|
7.0 | IC50 | 4 | — | |
JITAWAABXAQPMA
|
7.0 | IC50 | 4 | — | |
JKSGRMDJMCJGOZ
|
7.0 | IC50 | 4 | — |