Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODSKPPKANDQVKC
|
7.8 | IC50 | 2 | — | |
IWFSHKKFDSWNLZ
|
7.8 | IC50 | 4 | — | |
PHZKSLPIUQGPAT
|
7.8 | IC50 | 2 | — | |
YEUDACDOZNWCHD
|
7.8 | IC50 | 3 | — | |
HIXUASWPIBRERF
|
7.7 | IC50 | 4 | — | |
INUJXODUXNNZGR
|
7.7 | IC50 | 2 | — | |
CBFWZXFLDBEITH
|
7.7 | IC50 | 2 | — | |
IAMXTOFVAQFWAG
|
7.7 | IC50 | 4 | — | |
GJIDOEDDEGPTSO
|
7.7 | IC50 | 4 | — | |
UTZSWEGCKNIASP
|
7.7 | IC50 | 4 | — | |
ZZYMTFSRMGVTHN
|
7.7 | IC50 | 4 | — | |
KCBUDEQNWMMDNP
|
7.6 | IC50 | 2 | — | |
RAPGJWJWLNLLJV
|
7.6 | IC50 | 4 | — | |
KIULKJPSEKEYSN
|
7.6 | IC50 | 2 | — | |
JFYSQOAWENSFOW
|
7.6 | IC50 | 2 | — | |
ZFFPYADDQAFCLV
|
7.5 | IC50 | 2 | — | |
ZSRDAOYQIHISJX
|
7.5 | IC50 | 4 | — | |
LHVPLZJQMAJVNH
|
7.5 | IC50 | 2 | — | |
ZBWLUANTWWXFAY
|
7.5 | IC50 | 4 | — | |
DXWBQRNOIBKCRS
|
7.5 | IC50 | 2 | — | |
SRCSURSLBOIZMP
|
7.5 | IC50 | 4 | — | |
RANQSIYIJYBQSV
|
7.5 | IC50 | 4 | — | |
XFKGXBZSDIBBEB
|
7.5 | IC50 | 3 | — | |
FFPAJRVVMQCSIS
|
7.4 | IC50 | 2 | — | |
LQYFSFPPMCUGJG
|
7.4 | IC50 | 2 | — | |
HBVWDHIDINQCFS
|
7.3 | IC50 | 2 | — | |
FKRPRKAKBURXTN
|
7.3 | IC50 | 4 | — | |
CAAKGPRIVJHBKP
|
7.2 | IC50 | 2 | — | |
UDNJJABYGHGSGZ
|
7.2 | IC50 | 2 | — | |
SRAUODURYYKAAX
|
7.2 | IC50 | 4 | — | |
WTNCKLVOKCXDAU
|
7.2 | IC50 | 4 | — | |
LYPDEIQDNUKHGB
|
7.2 | IC50 | 4 | — | |
XRMAIQZIMRILDM
|
7.2 | IC50 | 4 | — | |
DZNOYNAVIGLCIO
|
7.2 | IC50 | 4 | — | |
VDUOAOAXBCEYSN
|
7.1 | IC50 | 4 | — | |
JAXMQOAWBPDQGA
|
7.1 | IC50 | 4 | — | |
JAXMQOAWBPDQGA
|
7.1 | IC50 | 4 | — | |
NDRMBCNSTDAADS
|
7.1 | IC50 | 4 | — | |
CQPMMSAANJNLLH
|
7.1 | IC50 | 4 | — | |
DTDZLJHKVNTQGZ
|
7.1 | IC50 | 4 | — | |
LCGNLQSOSJFLKR
|
7.1 | IC50 | 4 | — | |
VRUHOUHYPBCHJF
|
7.1 | IC50 | 4 | — | |
BXOOMWSWLIGVOJ
|
7.1 | IC50 | 2 | — | |
XPOQCGFJEGWPCZ
|
7.1 | IC50 | 4 | — | |
CFKHTEWRARJPEJ
|
7.0 | IC50 | 4 | — | |
NZKPNEZKGRFGOJ
|
7.0 | IC50 | 2 | — | |
XTPBKJJFRXGTTG
|
7.0 | IC50 | 4 | — | |
LUUINHUULZHSSK
|
7.0 | IC50 | 4 | — | |
WFJUFNKDUQHULP
|
7.0 | IC50 | 4 | — | |
ADSGNVVPFOHZGF
|
7.0 | IC50 | 4 | — |