Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHKJWWUZGWZKLR
|
8.0 | IC50 | 4 | — | |
MUQIBOPZUADQEJ
|
8.0 | IC50 | 4 | — | |
MZYFUTAKZNZIFC
|
8.0 | IC50 | 4 | — | |
NMNWEMCMDINIHC
|
8.0 | IC50 | 4 | — | |
NOMZDPJQKXSYBL
|
8.0 | IC50 | 4 | — | |
NQONOXVHKBUDCJ
|
8.0 | IC50 | 4 | — | |
NRZIYNYUTWCLTI
|
8.0 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
8.0 | IC50 | 4 | — | |
OWRAVMYSMHRQCB
|
8.0 | IC50 | 4 | — | |
PIUXSBGKAMYRFN
|
8.0 | IC50 | 4 | — | |
PNMORMAFEGBQRP
|
8.0 | IC50 | 4 | — | |
QDUFKTLTZYIENB
|
8.0 | IC50 | 4 | — | |
SORDPRCCLIYEOW
|
8.0 | IC50 | 4 | — | |
TXGKWJJIRGPDPH
|
8.0 | IC50 | 2 | — | |
VIAHIHPQYRESAI
|
8.0 | IC50 | 2 | — | |
WAZLJFYXSGVHFD
|
8.0 | IC50 | 2 | — | |
WCUSMKPGBOFBGV
|
8.0 | IC50 | 4 | — | |
WSTDGQPPQBLXGN
|
8.0 | IC50 | 4 | — | |
XWHRRPRMSJTOHZ
|
8.0 | IC50 | 4 | — | |
YKCSCWCEGAZILJ
|
8.0 | IC50 | 4 | — | |
ZASAXBVGTTZXFX
|
8.0 | IC50 | 2 | — | |
ZQLXLPNBWGVBKS
|
8.0 | IC50 | 4 | — | |
GZZMQXYSLCBPEA
|
8.0 | IC50 | 2 | — | |
IMWJPROBNIHLGY
|
8.0 | IC50 | 2 | — | |
IWPKWWKRBABODH
|
8.0 | IC50 | 2 | — | |
KOCGTJLQXCDACS
|
8.0 | IC50 | 2 | — | |
NDRHAIXHZKANNH
|
8.0 | IC50 | 2 | — | |
QBALEQIKDARBEA
|
8.0 | IC50 | 2 | — | |
UXPMAKAPBDDECI
|
8.0 | IC50 | 2 | — | |
ZGBFBHGZYPWPCB
|
8.0 | IC50 | 2 | — | |
HISIRLJXUDBATG
|
7.9 | IC50 | 2 | — | |
SGASELFPTYBIAK
|
7.9 | IC50 | 2 | — | |
TTZRKWJEYFCHTK
|
7.9 | IC50 | 2 | — | |
XIFBJTVEBBPQIC
|
7.9 | IC50 | 2 | — | |
XJNFXLGERDKDHP
|
7.9 | IC50 | 2 | — | |
AFENDHSQQLGKNV
|
7.9 | IC50 | 2 | — | |
NGIKAUHCSTVPFD
|
7.9 | IC50 | 2 | — | |
QSBISIOFJGEMQH
|
7.9 | IC50 | 4 | — | |
ROTSUPQHTLQDLC
|
7.9 | IC50 | 2 | — | |
TXEIMOIOXUHDIC
|
7.9 | IC50 | 2 | — | |
DWFZVULACSFMRM
|
7.8 | IC50 | 2 | — | |
IWKOKHWJIQAIFO
|
7.8 | IC50 | 2 | — | |
QBABDPMKOQHCQH
|
7.8 | IC50 | 2 | — | |
BVQHFOQYLXZHKL
|
7.8 | IC50 | 2 | — | |
LDYGDXKFRFPMHL
|
7.8 | IC50 | 2 | — | |
NAYKFOMEZLGWOU
|
7.8 | IC50 | 4 | — | |
SOSHINBXLNHODF
|
7.8 | IC50 | 2 | — | |
WIVWGJJPMANMAK
|
7.8 | IC50 | 2 | — | |
BDPATPOFNBRCCT
|
7.8 | IC50 | 4 | — | |
NGUHGFKCQBKIGO
|
7.8 | IC50 | 4 | — |