Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBOGEDJQULJRGL
|
8.2 | IC50 | 2 | — | |
PNECHCFDYAQPCJ
|
8.2 | IC50 | 2 | — | |
QMVPFGNVCUNBET
|
8.2 | IC50 | 2 | — | |
RXEHIULELGCSKA
|
8.2 | IC50 | 2 | — | |
RXTXTYQPYKEVKE
|
8.2 | IC50 | 2 | — | |
SDYHYNUKUWSPFA
|
8.2 | IC50 | 2 | — | |
WWTSWYZIBLALNY
|
8.2 | IC50 | 2 | — | |
YXRUPTXNZBVUOR
|
8.2 | IC50 | 2 | — | |
ADUOVQPGZNRALP
|
8.1 | IC50 | 2 | — | |
AEYCQUQWVCEEHF
|
8.1 | IC50 | 2 | — | |
ALGJUBJEQALNFZ
|
8.1 | IC50 | 2 | — | |
BWUHGFBIGNESMO
|
8.1 | IC50 | 2 | — | |
CVORHJZOOUPQIJ
|
8.1 | IC50 | 2 | — | |
GXBGRQPGTWTRDX
|
8.1 | IC50 | 2 | — | |
MPCBDAXTWLZHRP
|
8.1 | IC50 | 2 | — | |
NRGNIIHTGVGFJI
|
8.1 | IC50 | 2 | — | |
PRPYEHYKSGYPEL
|
8.1 | IC50 | 2 | — | |
VHKGMHJQUFVXHX
|
8.1 | IC50 | 4 | — | |
VJKAEDZFTRJFHX
|
8.1 | IC50 | 2 | — | |
VVLCJIFBCLQQDO
|
8.1 | IC50 | 4 | — | |
XNQCEAYNRGEWSL
|
8.1 | IC50 | 2 | — | |
DMOZBAPKYVVXQZ
|
8.1 | IC50 | 4 | — | |
GBKZKQJKTYRPJY
|
8.1 | IC50 | 2 | — | |
GDMZIUSWFQWRIG
|
8.1 | IC50 | 2 | — | |
KJLPVUNMMFZOME
|
8.1 | IC50 | 2 | — | |
MAVPBBTWLNFYBD
|
8.1 | IC50 | 2 | — | |
OFYZSZNDKNYQID
|
8.1 | IC50 | 2 | — | |
NXCCFZKYCZDCMZ
|
8.0 | IC50 | 2 | — | |
AHRQOACXLIJBJW
|
8.0 | IC50 | 2 | — | |
AYFZHEZEOZYSCU
|
8.0 | IC50 | 4 | — | |
BTUIGZUKKUYDCL
|
8.0 | IC50 | 4 | — | |
CDPFOGAUJZJOMI
|
8.0 | IC50 | 4 | — | |
CIUWUQLNBYAGJI
|
8.0 | IC50 | 2 | — | |
CNHZQWRCJQVKTD
|
8.0 | IC50 | 4 | — | |
CYJUFMHEEQFJAT
|
8.0 | IC50 | 6 | — | |
CYNIOIPKRXVGHL
|
8.0 | IC50 | 4 | — | |
DAYXEKSRINKFFG
|
8.0 | IC50 | 4 | — | |
DITRKTDSBBBRRK
|
8.0 | IC50 | 4 | — | |
DJPJWMXWFDIMFG
|
8.0 | IC50 | 4 | — | |
DKUKWIVFZJMJFK
|
8.0 | IC50 | 4 | — | |
DZGHOLAHGUXCFV
|
8.0 | IC50 | 4 | — | |
GTPCNCNWJUFVEI
|
8.0 | IC50 | 4 | — | |
GXMWDEYADMNXAV
|
8.0 | IC50 | 4 | — | |
IDGBYHLKGFLWNN
|
8.0 | IC50 | 4 | — | |
IWABBCZYAFPJND
|
8.0 | IC50 | 4 | — | |
JBINHQWXUMEKRF
|
8.0 | IC50 | 4 | — | |
JGUPBZDFMCZRNA
|
8.0 | IC50 | 4 | — | |
JLWRTIPIGXDNEG
|
8.0 | IC50 | 4 | — | |
JQCGLHYCQOFWMG
|
8.0 | IC50 | 4 | — | |
LYYXPHCAXQDCNN
|
8.0 | IC50 | 4 | — |