Target Details
| UniProt AC | Q15119 |
|---|---|
| Gene Symbol | PDK2 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 493
- Clinical molecules 0
- Avg pChEMBL 7.13
KEGG Pathways (1)
Active Molecules (493)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OINIDTBTTIYZIO
|
6.0 | IC50 | 4 | — | |
PABSUYDXHABXPY
|
6.0 | IC50 | 4 | — | |
PAVCFPGEDQLOLY
|
6.0 | IC50 | 4 | — | |
PUHWWAJTHDKCGR
|
6.0 | IC50 | 4 | — | |
PWDYOVIZDCYFRZ
|
6.0 | IC50 | 4 | — | |
PXUOKRBBSRTUNE
|
6.0 | IC50 | 4 | — | |
PZPMTBAIXNMBME
|
6.0 | IC50 | 4 | — | |
QMXIGKOHRUDNMV
|
6.0 | IC50 | 4 | — | |
QPFCZCMRUOQZRG
|
6.0 | IC50 | 4 | — | |
QQMKDSHSGYQMOV
|
6.0 | IC50 | 4 | — | |
QTZREWXFIMJBHN
|
6.0 | IC50 | 4 | — | |
QXCUSMAHYXWCOF
|
6.0 | IC50 | 4 | — | |
RECOPQDOXFPBNE
|
6.0 | IC50 | 4 | — | |
RFGOESLFDUAMGB
|
6.0 | IC50 | 4 | — | |
RTVPWYJBMHEYTA
|
6.0 | IC50 | 4 | — | |
RWEVXAYNUMFKQD
|
6.0 | IC50 | 4 | — | |
SLUNFEBZDXASNJ
|
6.0 | IC50 | 4 | — | |
SVXHTPKAAXLDLX
|
6.0 | IC50 | 4 | — | |
SYPAMOJTLDNMQL
|
6.0 | IC50 | 4 | — | |
UDUFRUMXLFCNQN
|
6.0 | IC50 | 4 | — | |
UKVBAJDPXOGHTO
|
6.0 | IC50 | 4 | — | |
UUGBZZQAHRXVBV
|
6.0 | IC50 | 4 | — | |
UZZOOCJSVGDZPS
|
6.0 | IC50 | 4 | — | |
VAEZIOUPBWPWKT
|
6.0 | IC50 | 4 | — | |
VKRJGZNMDIROFE
|
6.0 | IC50 | 4 | — | |
VLHPKUJISXSNFG
|
6.0 | IC50 | 4 | — | |
WHGYCNIXXDEKMI
|
6.0 | IC50 | 4 | — | |
WILCKYMTSIVKIZ
|
6.0 | IC50 | 4 | — | |
WLNHFWZZOOBEHX
|
6.0 | IC50 | 4 | — | |
WLSKWMBVRHXLLG
|
6.0 | IC50 | 4 | — | |
WREUMGOBADOOMR
|
6.0 | IC50 | 4 | — | |
WVWGMHSCWFAKFO
|
6.0 | IC50 | 4 | — | |
WWCJRXYIKMLMHV
|
6.0 | IC50 | 4 | — | |
WYNUQGLAIYDBRL
|
6.0 | IC50 | 4 | — | |
XAWMWRRMUXYKPC
|
6.0 | IC50 | 4 | — | |
XDDFKFMQTWAHQW
|
6.0 | IC50 | 4 | — | |
XOEWAGGFKMWDPJ
|
6.0 | IC50 | 4 | — | |
YASUGMSGTIVYCC
|
6.0 | IC50 | 4 | — | |
YAYMVYXCAZWMFA
|
6.0 | IC50 | 4 | — | |
YZZSZNYNWZBIOJ
|
6.0 | IC50 | 4 | — | |
ZBEYKNGCVKIDQV
|
6.0 | IC50 | 4 | — | |
ZRJGAZHGDXMXNT
|
6.0 | IC50 | 4 | — | |
ZWUZKCPHVDLAAI
|
6.0 | IC50 | 4 | — |