Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTSYVKWXYINLJV
|
6.5 | IC50 | 4 | — | |
ZWUZKCPHVDLAAI
|
6.5 | IC50 | 4 | — | |
AUJRIOZTXXHUGR
|
6.5 | IC50 | 4 | — | |
BQRFDZQRKCARHX
|
6.5 | IC50 | 4 | — | |
BTVCELJQYVYBMY
|
6.5 | IC50 | 4 | — | |
DXULLUCLDXLAEE
|
6.5 | IC50 | 4 | — | |
FBRKPMZCQHNIJI
|
6.5 | IC50 | 4 | — | |
FKHMXABMILEREF
|
6.5 | IC50 | 4 | — | |
GNIVANXSNOBJOV
|
6.5 | IC50 | 4 | — | |
HJCYHYZYHRDVBU
|
6.5 | IC50 | 4 | — | |
HSRXRPVIBOXEKS
|
6.5 | IC50 | 4 | — | |
KCXGMKDIPWGLSK
|
6.5 | IC50 | 4 | — | |
KHWHZLYCFONFBB
|
6.5 | IC50 | 4 | — | |
KURLHYDERFSDAV
|
6.5 | IC50 | 4 | — | |
KUUZLDUCOUHSFK
|
6.5 | IC50 | 4 | — | |
LNBYJUPTVFIGQB
|
6.5 | IC50 | 4 | — | |
MTLYSRUJNCWFOX
|
6.5 | IC50 | 4 | — | |
PABSUYDXHABXPY
|
6.5 | IC50 | 4 | — | |
PYWNULWLMYXJIE
|
6.5 | IC50 | 4 | — | |
QWHBUKMSQWNPLU
|
6.5 | IC50 | 4 | — | |
REKSHMUIHDBZEL
|
6.5 | IC50 | 4 | — | |
UHLKSPFADXABBK
|
6.5 | IC50 | 4 | — | |
UKVBAJDPXOGHTO
|
6.5 | IC50 | 4 | — | |
VKRJGZNMDIROFE
|
6.5 | IC50 | 4 | — | |
WQBUEPUJTZXCSW
|
6.5 | IC50 | 4 | — | |
WYUKVGVZYSCCDJ
|
6.5 | IC50 | 4 | — | |
XXFAGYMXMCJALN
|
6.5 | IC50 | 4 | — | |
XZGKZXADQIAIAB
|
6.5 | IC50 | 4 | — | |
ZQLXLPNBWGVBKS
|
6.5 | IC50 | 4 | — | |
MZIWZDMEFARRSI
|
6.5 | IC50 | 2 | — | |
JKJOXJGLLJZNII
|
6.4 | IC50 | 2 | — | |
AFZSMODLJJCVPP
|
6.4 | IC50 | 12 | — | |
LHSKWVQEAJUPOG
|
6.4 | IC50 | 4 | — | |
OVUREOQFPBNHNM
|
6.4 | IC50 | 4 | — | |
DLCOOKRUECVLCI
|
6.4 | IC50 | 3 | — | |
UKBGBACORPRCGG
|
6.4 | IC50 | 17 | — | |
XCPMMIISBZJPHR
|
6.4 | IC50 | 3 | — | |
KLYXBLDJCZSBIR
|
6.3 | IC50 | 2 | — | |
YJJKWAZEMDORLO
|
6.3 | IC50 | 3 | — | |
WHBHHAKSCKVYCJ
|
6.3 | IC50 | 3 | — | |
ZPJHXZDMLBZMJK
|
6.3 | IC50 | 3 | — | |
RPNZGGQCZUXPBC
|
6.2 | IC50 | 4 | — | |
QWXFJSQDZDYGBJ
|
6.2 | IC50 | 3 | — | |
NLHSXYGKBUOFPL
|
6.2 | IC50 | 4 | — | |
SICRPGFNFVPIKM
|
6.2 | IC50 | 3 | — | |
ZYLHCSSOEGIFAO
|
6.2 | IC50 | 3 | — | |
ORWIYCURPDKSBI
|
6.1 | IC50 | 15 | Yes | |
YPRFHQADDZVCKY
|
6.1 | IC50 | 3 | — | |
OWXORKPNCHJYOF
|
6.1 | IC50 | 17 | Yes | |
JAOFIBKJPAHQNQ
|
6.1 | IC50 | 4 | — |