Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YZZSZNYNWZBIOJ
|
7.0 | IC50 | 4 | — | |
ZBEYKNGCVKIDQV
|
7.0 | IC50 | 4 | — | |
ZPMRFYJDPARNBL
|
7.0 | IC50 | 4 | — | |
ZUZGRFYAGRDPGJ
|
7.0 | IC50 | 4 | — | |
ZVFIHSAIQWKOAE
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZXOPKIJCZPLJBU
|
7.0 | IC50 | 4 | — | |
ZYAAUDLDGUEAPN
|
7.0 | IC50 | 4 | — | |
ZYLSRWYAGYUONP
|
7.0 | IC50 | 4 | — | |
BGFOEUFOBZQIEL
|
7.0 | IC50 | 2 | — | |
HJUAIOQSNLTXLS
|
7.0 | IC50 | 2 | — | |
CJKPVNLQNOSPAE
|
7.0 | IC50 | 4 | — | |
CYNYZDWGNQYJDF
|
7.0 | IC50 | 3 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
MUBBTSZWDVFVLT
|
7.0 | IC50 | 3 | — | |
URBQRLTYIDBJQO
|
7.0 | IC50 | 4 | — | |
FSMLYTJJLFECDK
|
7.0 | IC50 | 4 | — | |
TYTXGPAMIGYEGN
|
7.0 | IC50 | 4 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
ZWUKNHQASDKHCT
|
6.9 | IC50 | 4 | — | |
KOAXITXTHITWLT
|
6.9 | IC50 | 4 | — | |
KDSTWUUMLDUNDV
|
6.9 | IC50 | 3 | — | |
NSEKNXMDWSTZJL
|
6.9 | IC50 | 4 | — | |
XNGVNSXRRADPSC
|
6.9 | IC50 | 4 | — | |
RXSXHCNTLOATRW
|
6.9 | Ki | 2 | — | |
XLFNLJYGUOLEJS
|
6.9 | IC50 | 26 | — | |
BUUKMYSHPSEDRR
|
6.9 | IC50 | 2 | — | |
ZPNZQVNPYMEKML
|
6.9 | IC50 | 4 | — | |
TWRWVLYTPAORIW
|
6.8 | IC50 | 4 | — | |
VPETUWRKODTKNY
|
6.8 | IC50 | 4 | — | |
ZBCASIFBVICMSH
|
6.8 | IC50 | 4 | — | |
KHPDVVDNRUBARQ
|
6.8 | IC50 | 2 | — | |
CWHNQKPCYFFKDR
|
6.8 | IC50 | 4 | — | |
FLCLKDRMVXBLHR
|
6.8 | IC50 | 4 | — | |
IXYGIIBGSMZJMY
|
6.8 | IC50 | 3 | — | |
KKVYOWPPMNSLCP
|
6.8 | IC50 | 5 | — | |
ZOPYDEDEHVUGTC
|
6.8 | IC50 | 4 | — | |
BQKIJENXHZFRRG
|
6.8 | IC50 | 3 | — | |
LDFLSIZNFQLCDQ
|
6.8 | IC50 | 4 | — | |
GFICNEUSPWSTPP
|
6.8 | IC50 | 4 | — | |
MJTMTQQRDNWPGK
|
6.7 | Ki | 4 | — | |
USCKZBKHRWIQAC
|
6.7 | IC50 | 3 | — | |
HVZAUSYZLGXKIP
|
6.7 | IC50 | 4 | — | |
QRPZFMFZNJHOTN
|
6.6 | IC50 | 4 | — | |
GAFYAXXDUJHTEI
|
6.6 | IC50 | 4 | — | |
WSCBMCCISYODBR
|
6.6 | IC50 | 3 | — | |
YJCWUJKWNBKVAH
|
6.6 | IC50 | 2 | — | |
YJJQLXIDSMWSDE
|
6.6 | Ki | 2 | — | |
QTZREWXFIMJBHN
|
6.5 | IC50 | 4 | — | |
XJVOPOWBIDUKFI
|
6.5 | IC50 | 4 | — |