Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OYIVLQTWURCFIL
|
7.0 | IC50 | 4 | — | |
OYIVLQTWURCFIL
|
7.0 | IC50 | 4 | — | |
OZPNMFRXHFNHAE
|
7.0 | IC50 | 4 | — | |
PAVCFPGEDQLOLY
|
7.0 | IC50 | 4 | — | |
PRCTUAYWNHMKTR
|
7.0 | IC50 | 4 | — | |
PSQMYJVREYGDAB
|
7.0 | IC50 | 4 | — | |
PTHJRVBBACHGOH
|
7.0 | IC50 | 4 | — | |
PUPFOOFVPKXKKS
|
7.0 | IC50 | 4 | — | |
QAAAEMHGCDUTQF
|
7.0 | IC50 | 4 | — | |
QEHFXBQCHXZVPP
|
7.0 | IC50 | 4 | — | |
QMXIGKOHRUDNMV
|
7.0 | IC50 | 4 | — | |
QOBHBSIALHUBML
|
7.0 | IC50 | 4 | — | |
QOMVKWOSNCOMEE
|
7.0 | IC50 | 4 | — | |
QORZJUPQLUQVLM
|
7.0 | IC50 | 4 | — | |
QPFCZCMRUOQZRG
|
7.0 | IC50 | 4 | — | |
QQEXAKLRPMBVMU
|
7.0 | IC50 | 4 | — | |
QVSHTTDOPIXQHK
|
7.0 | IC50 | 4 | — | |
RRPLLQMMPJWFIR
|
7.0 | IC50 | 4 | — | |
RRVGEDSKKYXEEQ
|
7.0 | IC50 | 4 | — | |
RWEVXAYNUMFKQD
|
7.0 | IC50 | 4 | — | |
RWKAWUMWADJEBW
|
7.0 | IC50 | 4 | — | |
SJEXWLLUJGZGAK
|
7.0 | IC50 | 4 | — | |
SQEBZRWBDVPJDR
|
7.0 | IC50 | 4 | — | |
SWUFKVPRVHWIRW
|
7.0 | IC50 | 4 | — | |
SXBULXXRUIFERC
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
SZCHNEBNXWTYGU
|
7.0 | IC50 | 4 | — | |
TZKXWAODTKIRQH
|
7.0 | IC50 | 4 | — | |
UDXRPQUWDSCOTK
|
7.0 | IC50 | 4 | — | |
UMRLOUSNWOYFFM
|
7.0 | IC50 | 4 | — | |
UOLOUISPBSPRGG
|
7.0 | IC50 | 4 | — | |
VIRNQTUQCWCOAV
|
7.0 | IC50 | 4 | — | |
VLTVCXJATKADNO
|
7.0 | IC50 | 4 | — | |
VPMACFXFRUVPQK
|
7.0 | IC50 | 4 | — | |
WBZWNTJAWZVNCI
|
7.0 | IC50 | 4 | — | |
WEJYENUPPGWUCM
|
7.0 | IC50 | 4 | — | |
WEWLWBDTDINJNR
|
7.0 | IC50 | 4 | — | |
WKTAYYWOLXTJGL
|
7.0 | IC50 | 4 | — | |
WQJHFNBULHHCAT
|
7.0 | IC50 | 4 | — | |
XBXCLVBYMZQBFQ
|
7.0 | IC50 | 4 | — | |
XNWFFSUKXSXYOJ
|
7.0 | IC50 | 4 | — | |
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XRQPVXUTZFDCGK
|
7.0 | IC50 | 4 | — | |
XVLUOKHYAJARDM
|
7.0 | IC50 | 4 | — | |
YDTBZYAJXNXQGG
|
7.0 | IC50 | 4 | — | |
YKCSCWCEGAZILJ
|
7.0 | IC50 | 4 | — | |
YQIDANKABBOUGC
|
7.0 | IC50 | 4 | — | |
YTDJEAZYTGIAJJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — | |
YZOMOQFRSNGZMJ
|
7.0 | IC50 | 4 | — |