Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVWCFDQTLRXQFX
|
7.0 | IC50 | 4 | — | |
GAEIKTXZNLANQY
|
7.0 | IC50 | 4 | — | |
GIFBFVKPOAPOQF
|
7.0 | IC50 | 4 | — | |
GOYZFCBIPVDHLA
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
GRGOYLVPZGFXOI
|
7.0 | IC50 | 4 | — | |
HBQAMWIICPEKLM
|
7.0 | IC50 | 4 | — | |
HEZXCHOQRVOWOO
|
7.0 | IC50 | 4 | — | |
HMDVVVVFTDRVEN
|
7.0 | IC50 | 4 | — | |
HOTHCUMDFKWXAY
|
7.0 | IC50 | 4 | — | |
HPKSWZBPOBFFGH
|
7.0 | IC50 | 4 | — | |
HQXGHFGYLLOUQN
|
7.0 | IC50 | 4 | — | |
HUZNUFRXRYRKLQ
|
7.0 | IC50 | 4 | — | |
HXGAMFVEHXJPPA
|
7.0 | IC50 | 4 | — | |
IAOKECPRCAJJLW
|
7.0 | IC50 | 4 | — | |
IBOAFKTZBFJUKA
|
7.0 | IC50 | 4 | — | |
IJYGCXRXUFNBBX
|
7.0 | IC50 | 4 | — | |
JEULTWLFDMZUPQ
|
7.0 | IC50 | 4 | — | |
JITAWAABXAQPMA
|
7.0 | IC50 | 4 | — | |
JKSGRMDJMCJGOZ
|
7.0 | IC50 | 4 | — | |
JLVBJWREILIRAS
|
7.0 | IC50 | 4 | — | |
JLWPPFZGJGHSTJ
|
7.0 | IC50 | 4 | — | |
JMIVUIMGDJZLIG
|
7.0 | IC50 | 4 | — | |
JNGRLPFNEIFOTG
|
7.0 | IC50 | 4 | — | |
JOCFMBDFPBFGGL
|
7.0 | IC50 | 4 | — | |
JOJIFEAFJOWRTN
|
7.0 | IC50 | 4 | — | |
KLQHYYHEUCEROZ
|
7.0 | IC50 | 4 | — | |
KLQHYYHEUCEROZ
|
7.0 | IC50 | 4 | — | |
KZUMTKNLJKJSBD
|
7.0 | IC50 | 4 | — | |
KZUMTKNLJKJSBD
|
7.0 | IC50 | 4 | — | |
LKBFKOYSSYSDQH
|
7.0 | IC50 | 4 | — | |
LLGHHTDOUJTEOP
|
7.0 | IC50 | 4 | — | |
LLWJFRPCKCAMKV
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LRFWDRILVLEZJM
|
7.0 | IC50 | 4 | — | |
LSJRQFSUVPSXTH
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
LWPVJGVLNMPBPK
|
7.0 | IC50 | 4 | — | |
MJDOETCLTIAWPE
|
7.0 | IC50 | 4 | — | |
MMIWOBFOVOZMKG
|
7.0 | IC50 | 4 | — | |
MMWXYJPJGRRGIT
|
7.0 | IC50 | 4 | — | |
NDZDDEMSENNYBA
|
7.0 | IC50 | 4 | — | |
NEXLZTATSAIBTR
|
7.0 | IC50 | 4 | — | |
NMNWEMCMDINIHC
|
7.0 | IC50 | 4 | — | |
NSMJZJFXYGOOET
|
7.0 | IC50 | 4 | — | |
OAODSMWKFRASCR
|
7.0 | IC50 | 4 | — | |
OCVNXALHQSJRLS
|
7.0 | IC50 | 4 | — | |
OFVWPLPGVMYLFN
|
7.0 | IC50 | 4 | — | |
OJZZFYPZMQVSJV
|
7.0 | IC50 | 4 | — | |
OWFZQPQOHDKLNC
|
7.0 | IC50 | 4 | — |