Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VAVXGGRQQJZYBL
|
7.2 | IC50 | 8 | — | |
HBVWDHIDINQCFS
|
7.2 | IC50 | 2 | — | |
IWFSHKKFDSWNLZ
|
7.2 | IC50 | 4 | — | |
XRMAIQZIMRILDM
|
7.2 | IC50 | 4 | — | |
FIDDBBSOQKUFGA
|
7.2 | IC50 | 3 | — | |
SFQMDVJNIAAAJA
|
7.2 | IC50 | 4 | — | |
XFKGXBZSDIBBEB
|
7.2 | IC50 | 3 | — | |
DZNOYNAVIGLCIO
|
7.2 | IC50 | 4 | — | |
VDUOAOAXBCEYSN
|
7.1 | IC50 | 4 | — | |
JAXMQOAWBPDQGA
|
7.1 | IC50 | 4 | — | |
JAXMQOAWBPDQGA
|
7.1 | IC50 | 4 | — | |
NDRMBCNSTDAADS
|
7.1 | IC50 | 4 | — | |
CQPMMSAANJNLLH
|
7.1 | IC50 | 4 | — | |
VRUHOUHYPBCHJF
|
7.1 | IC50 | 4 | — | |
XPOQCGFJEGWPCZ
|
7.1 | IC50 | 4 | — | |
CFKHTEWRARJPEJ
|
7.0 | IC50 | 4 | — | |
ILEZYMARHZUBGD
|
7.0 | IC50 | 2 | — | |
MJTMTQQRDNWPGK
|
7.0 | Ki | 4 | — | |
WFJUFNKDUQHULP
|
7.0 | IC50 | 4 | — | |
ADSGNVVPFOHZGF
|
7.0 | IC50 | 4 | — | |
ADYFSAHHBUQVGK
|
7.0 | IC50 | 4 | — | |
AEROUCXDUDYEKO
|
7.0 | IC50 | 4 | — | |
AGIRAUWGTYSFEY
|
7.0 | IC50 | 4 | — | |
APWMGNIAYJJUAF
|
7.0 | IC50 | 4 | — | |
ARUCEZREJLJFDT
|
7.0 | IC50 | 4 | — | |
BCJWSMLGFKGOGY
|
7.0 | IC50 | 4 | — | |
BEDBXCKARVIOCD
|
7.0 | IC50 | 4 | — | |
BPZOUMFIFRETCA
|
7.0 | IC50 | 4 | — | |
BQUDNQLXMYGDNQ
|
7.0 | IC50 | 4 | — | |
BSLIZBUPULPNHQ
|
7.0 | IC50 | 4 | — | |
BSLIZBUPULPNHQ
|
7.0 | IC50 | 4 | — | |
BSQGGNPQVHKELV
|
7.0 | IC50 | 4 | — | |
BYSDPXBOYDDWFZ
|
7.0 | IC50 | 4 | — | |
CAIPBEZKRVGEKE
|
7.0 | IC50 | 4 | — | |
CGIKZEQNOIDVOV
|
7.0 | IC50 | 4 | — | |
CGYZWZHPCJOISU
|
7.0 | IC50 | 4 | — | |
CGYZWZHPCJOISU
|
7.0 | IC50 | 4 | — | |
CHWXLTDPQZWFAM
|
7.0 | IC50 | 4 | — | |
CXYRJLAOPDAFSS
|
7.0 | IC50 | 4 | — | |
CXYRJLAOPDAFSS
|
7.0 | IC50 | 4 | — | |
CYESLTXMVJMIOU
|
7.0 | IC50 | 4 | — | |
DGUGNQFTCBUBEL
|
7.0 | IC50 | 4 | — | |
DTLSNWXWIAFKCH
|
7.0 | IC50 | 4 | — | |
FBLPPJHSHGACEJ
|
7.0 | IC50 | 4 | — | |
FHANGEZWICYMAN
|
7.0 | IC50 | 4 | — | |
FHCJWURPGGJVIU
|
7.0 | IC50 | 4 | — | |
FLMXFYUZYPWMHO
|
7.0 | IC50 | 4 | — | |
FPKYIUHRFOETKG
|
7.0 | IC50 | 4 | — | |
FUJJLTFFZUJRAF
|
7.0 | IC50 | 4 | — | |
FURRPKJZBWBALL
|
7.0 | IC50 | 4 | — |