Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BDPATPOFNBRCCT
|
7.8 | IC50 | 4 | — | |
NGUHGFKCQBKIGO
|
7.8 | IC50 | 4 | — | |
QBABDPMKOQHCQH
|
7.8 | IC50 | 2 | — | |
XFLXHBRVXWEPCZ
|
7.8 | IC50 | 4 | — | |
YEUDACDOZNWCHD
|
7.8 | IC50 | 3 | — | |
LHVPLZJQMAJVNH
|
7.8 | IC50 | 2 | — | |
YDCQPNSQDQCBFM
|
7.8 | IC50 | 3 | — | |
IAMXTOFVAQFWAG
|
7.7 | IC50 | 4 | — | |
CBFWZXFLDBEITH
|
7.7 | IC50 | 2 | — | |
GJIDOEDDEGPTSO
|
7.7 | IC50 | 4 | — | |
LYPDEIQDNUKHGB
|
7.7 | IC50 | 4 | — | |
NGIKAUHCSTVPFD
|
7.7 | IC50 | 2 | — | |
RTYCQDBBCMTUFF
|
7.7 | IC50 | 4 | — | |
SOVOJYOIAXOTIM
|
7.7 | IC50 | 3 | — | |
UTZSWEGCKNIASP
|
7.7 | IC50 | 4 | — | |
ZZYMTFSRMGVTHN
|
7.7 | IC50 | 4 | — | |
RAPGJWJWLNLLJV
|
7.6 | IC50 | 4 | — | |
OXQTXJIDMWRZLX
|
7.6 | IC50 | 4 | — | |
VJSMYBWGSKJUEL
|
7.6 | IC50 | 4 | — | |
FOFVZTDYBUEDIT
|
7.6 | IC50 | 3 | — | |
KCBUDEQNWMMDNP
|
7.6 | IC50 | 2 | — | |
ZHMRBKJCNFNYIU
|
7.5 | IC50 | 3 | — | |
LQYFSFPPMCUGJG
|
7.5 | IC50 | 2 | — | |
ZSRDAOYQIHISJX
|
7.5 | IC50 | 4 | — | |
GLYKHSDGYVKDPV
|
7.5 | IC50 | 3 | — | |
IRGFJNBJMFGIAK
|
7.5 | IC50 | 4 | — | |
LSEQOPAXXJYNDG
|
7.5 | IC50 | 4 | — | |
QTUKYQAPKFQRDT
|
7.5 | IC50 | 4 | — | |
ZBWLUANTWWXFAY
|
7.5 | IC50 | 4 | — | |
SRCSURSLBOIZMP
|
7.5 | IC50 | 4 | — | |
RANQSIYIJYBQSV
|
7.5 | IC50 | 4 | — | |
CYJUFMHEEQFJAT
|
7.4 | IC50 | 6 | — | |
KIULKJPSEKEYSN
|
7.4 | IC50 | 2 | — | |
DTDZLJHKVNTQGZ
|
7.4 | IC50 | 4 | — | |
FFPAJRVVMQCSIS
|
7.4 | IC50 | 2 | — | |
HIXUASWPIBRERF
|
7.4 | IC50 | 4 | — | |
LCGNLQSOSJFLKR
|
7.4 | IC50 | 4 | — | |
INUJXODUXNNZGR
|
7.3 | IC50 | 2 | — | |
FKRPRKAKBURXTN
|
7.3 | IC50 | 4 | — | |
LZCHVMYGVHFFSN
|
7.3 | IC50 | 6 | — | |
DXWBQRNOIBKCRS
|
7.3 | IC50 | 2 | — | |
ZFFPYADDQAFCLV
|
7.3 | IC50 | 2 | — | |
XONRTPBYDAFIRW
|
7.3 | IC50 | 9 | — | |
UFRHUTDVBLSOCA
|
7.3 | IC50 | 2 | — | |
AQFMGFCVDBEMQE
|
7.2 | IC50 | 3 | — | |
XTPBKJJFRXGTTG
|
7.2 | IC50 | 4 | — | |
YXMBLKCXYORPJJ
|
7.2 | IC50 | 3 | — | |
SRAUODURYYKAAX
|
7.2 | IC50 | 4 | — | |
JFYSQOAWENSFOW
|
7.2 | IC50 | 2 | — | |
WTNCKLVOKCXDAU
|
7.2 | IC50 | 4 | — |