Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNHZQWRCJQVKTD
|
8.0 | IC50 | 4 | — | |
CYNIOIPKRXVGHL
|
8.0 | IC50 | 4 | — | |
DAYXEKSRINKFFG
|
8.0 | IC50 | 4 | — | |
DITRKTDSBBBRRK
|
8.0 | IC50 | 4 | — | |
DJPJWMXWFDIMFG
|
8.0 | IC50 | 4 | — | |
DKUKWIVFZJMJFK
|
8.0 | IC50 | 4 | — | |
DZGHOLAHGUXCFV
|
8.0 | IC50 | 4 | — | |
GTPCNCNWJUFVEI
|
8.0 | IC50 | 4 | — | |
GXMWDEYADMNXAV
|
8.0 | IC50 | 4 | — | |
IDGBYHLKGFLWNN
|
8.0 | IC50 | 4 | — | |
IWABBCZYAFPJND
|
8.0 | IC50 | 4 | — | |
JBINHQWXUMEKRF
|
8.0 | IC50 | 4 | — | |
JGUPBZDFMCZRNA
|
8.0 | IC50 | 4 | — | |
JLWRTIPIGXDNEG
|
8.0 | IC50 | 4 | — | |
JQCGLHYCQOFWMG
|
8.0 | IC50 | 4 | — | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
LYYXPHCAXQDCNN
|
8.0 | IC50 | 4 | — | |
MHKJWWUZGWZKLR
|
8.0 | IC50 | 4 | — | |
MUQIBOPZUADQEJ
|
8.0 | IC50 | 4 | — | |
MZYFUTAKZNZIFC
|
8.0 | IC50 | 4 | — | |
NMNWEMCMDINIHC
|
8.0 | IC50 | 4 | — | |
NOMZDPJQKXSYBL
|
8.0 | IC50 | 4 | — | |
NQONOXVHKBUDCJ
|
8.0 | IC50 | 4 | — | |
NRZIYNYUTWCLTI
|
8.0 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
8.0 | IC50 | 4 | — | |
OWRAVMYSMHRQCB
|
8.0 | IC50 | 4 | — | |
PIUXSBGKAMYRFN
|
8.0 | IC50 | 4 | — | |
PNMORMAFEGBQRP
|
8.0 | IC50 | 4 | — | |
QDUFKTLTZYIENB
|
8.0 | IC50 | 4 | — | |
SORDPRCCLIYEOW
|
8.0 | IC50 | 4 | — | |
TXEIMOIOXUHDIC
|
8.0 | IC50 | 2 | — | |
WAZLJFYXSGVHFD
|
8.0 | IC50 | 2 | — | |
WCUSMKPGBOFBGV
|
8.0 | IC50 | 4 | — | |
WSTDGQPPQBLXGN
|
8.0 | IC50 | 4 | — | |
XWHRRPRMSJTOHZ
|
8.0 | IC50 | 4 | — | |
YKCSCWCEGAZILJ
|
8.0 | IC50 | 4 | — | |
ZQLXLPNBWGVBKS
|
8.0 | IC50 | 4 | — | |
AHRQOACXLIJBJW
|
8.0 | IC50 | 2 | — | |
IMWJPROBNIHLGY
|
8.0 | IC50 | 2 | — | |
CIUWUQLNBYAGJI
|
7.9 | IC50 | 2 | — | |
ODSKPPKANDQVKC
|
7.9 | IC50 | 2 | — | |
WIVWGJJPMANMAK
|
7.9 | IC50 | 2 | — | |
HISIRLJXUDBATG
|
7.9 | IC50 | 2 | — | |
QSBISIOFJGEMQH
|
7.9 | IC50 | 4 | — | |
VIAHIHPQYRESAI
|
7.9 | IC50 | 2 | — | |
LDYGDXKFRFPMHL
|
7.8 | IC50 | 2 | — | |
LUUINHUULZHSSK
|
7.8 | IC50 | 4 | — | |
OFYZSZNDKNYQID
|
7.8 | IC50 | 2 | — | |
NAYKFOMEZLGWOU
|
7.8 | IC50 | 4 | — | |
NULXZQHTQSFRHZ
|
7.8 | IC50 | 4 | — |