Target Details
| UniProt AC | Q15118 |
|---|---|
| Gene Symbol | PDK1 |
| Protein Name | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10436 (BCDHK_Adom3) PF02518 (HATPase_c) |
Summary
- Multi-target molecules 524
- Clinical molecules 3
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (524)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RVFAVDLRKCTLLH
|
8.3 | IC50 | 2 | — | |
UXPMAKAPBDDECI
|
8.3 | IC50 | 2 | — | |
WWTSWYZIBLALNY
|
8.3 | IC50 | 2 | — | |
YXBMUKIETBHKNP
|
8.3 | IC50 | 2 | — | |
ZKIGCOOJJXCDGU
|
8.3 | IC50 | 2 | — | |
KNPYQCPWTWANOG
|
8.2 | IC50 | 2 | — | |
ALGJUBJEQALNFZ
|
8.2 | IC50 | 2 | — | |
BIFLYFTZKFZUAU
|
8.2 | IC50 | 2 | — | |
BWUHGFBIGNESMO
|
8.2 | IC50 | 2 | — | |
COPUGPVQCHSAPU
|
8.2 | IC50 | 2 | — | |
DRPJZMIFBAXAKX
|
8.2 | IC50 | 3 | — | |
GBKZKQJKTYRPJY
|
8.2 | IC50 | 2 | — | |
KJLPVUNMMFZOME
|
8.2 | IC50 | 2 | — | |
KOCGTJLQXCDACS
|
8.2 | IC50 | 2 | — | |
NRGNIIHTGVGFJI
|
8.2 | IC50 | 2 | — | |
NYDJCHUCGSSLJH
|
8.2 | IC50 | 2 | — | |
PCIALRSXUYBERL
|
8.2 | IC50 | 2 | — | |
QBALEQIKDARBEA
|
8.2 | IC50 | 2 | — | |
RXTXTYQPYKEVKE
|
8.2 | IC50 | 2 | — | |
SGASELFPTYBIAK
|
8.2 | IC50 | 2 | — | |
SOSHINBXLNHODF
|
8.2 | IC50 | 2 | — | |
TTZRKWJEYFCHTK
|
8.2 | IC50 | 2 | — | |
AFENDHSQQLGKNV
|
8.2 | IC50 | 2 | — | |
HNXNABSRTQYJCK
|
8.2 | IC50 | 2 | — | |
IWKOKHWJIQAIFO
|
8.2 | IC50 | 2 | — | |
MAVPBBTWLNFYBD
|
8.2 | IC50 | 2 | — | |
MWGZGIZAANWRLL
|
8.2 | IC50 | 4 | — | |
YXRUPTXNZBVUOR
|
8.2 | IC50 | 2 | — | |
ZGBFBHGZYPWPCB
|
8.2 | IC50 | 2 | — | |
CBIRAASKUXNRFE
|
8.1 | IC50 | 2 | — | |
CVORHJZOOUPQIJ
|
8.1 | IC50 | 2 | — | |
NDRHAIXHZKANNH
|
8.1 | IC50 | 2 | — | |
TXGKWJJIRGPDPH
|
8.1 | IC50 | 2 | — | |
VVLCJIFBCLQQDO
|
8.1 | IC50 | 4 | — | |
XIFBJTVEBBPQIC
|
8.1 | IC50 | 2 | — | |
XJNFXLGERDKDHP
|
8.1 | IC50 | 2 | — | |
ZASAXBVGTTZXFX
|
8.1 | IC50 | 2 | — | |
DMOZBAPKYVVXQZ
|
8.1 | IC50 | 4 | — | |
XLYVQVWMTOLDNL
|
8.1 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
8.1 | IC50 | 21 | — | |
AEYCQUQWVCEEHF
|
8.1 | IC50 | 2 | — | |
DWFZVULACSFMRM
|
8.1 | IC50 | 2 | — | |
IWPKWWKRBABODH
|
8.1 | IC50 | 2 | — | |
PRPYEHYKSGYPEL
|
8.1 | IC50 | 2 | — | |
ROTSUPQHTLQDLC
|
8.1 | IC50 | 2 | — | |
VHKGMHJQUFVXHX
|
8.1 | IC50 | 4 | — | |
VJKAEDZFTRJFHX
|
8.1 | IC50 | 2 | — | |
AYFZHEZEOZYSCU
|
8.0 | IC50 | 4 | — | |
BTUIGZUKKUYDCL
|
8.0 | IC50 | 4 | — | |
CDPFOGAUJZJOMI
|
8.0 | IC50 | 4 | — |